SCHEMBL9921580

SCHEMBL9921580

CN1CCC([N+](=O)[O-])([N+](=O)[O-])CC1

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NEK2 P51955 1/20 0.38
SIRT6 Q8N6T7 1/20 0.35
GAA P10253 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
LMNA P02545 1/20 0.32
ALDH1A1 P00352 1/20 0.32
HPGD P15428 1/20 0.32
CRHBP P24387 1/20 0.31
CRHR2 Q13324 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9947431 0.88 NEK2 (0.34) NEK2SIRT6GAACRHBPCRHR2
SCHEMBL27734250 0.78 L3MBTL1 (0.33) NEK2SIRT6GAAL3MBTL1ALDH1A1
Methane SCHEMBL27480548 0.77 L3MBTL1 (0.32) SIRT6GAAL3MBTL1ALDH1A1HPGD
SCHEMBL9918124 0.77 CYP2D6 (0.37) GAALMNAALDH1A1
SCHEMBL14911002 0.76
SCHEMBL9921596 0.76 GAA (0.38) SIRT6GAAALDH1A1CRHBPCRHR2
SCHEMBL28392433 0.71 NLRP3 (0.33)
SCHEMBL3285840 0.71 NLRP3 (0.33)
SCHEMBL25475858 0.69 CRHBP (0.50) GAACRHBPCRHR2
SCHEMBL3289507 0.69 NLRP3 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20140308260-A1 METHODS AND COMPOSITIONS COMPRISING A NITRITE-REDUCTASE PROMOTER FOR TREATMENT OF MEDICAL DISORDERS AND PRESERVATION OF BLOOD PRODUCTS EPICENTRX, INC. 2014-10-16 US disclosed
WO-2013052803-A2 METHODS AND COMPOSITIONS COMPRISING A NITRITE-REDUCTASE PROMOTER FOR TREATMENT OF MEDICAL DISORDERS AND PRESERVATION OF BLOOD PRODUCTS RADIORX, INC. (US) 2013-04-11 WO disclosed
US-20120149678-A1 Organonitro Compounds for Use in Treating Non-Hodgkin's Lymphoma and Leukemia, and Methods Relating Thereto ORONSKY BRYAN T (US) 2012-06-14 US disclosed
WO-2012078992-A1 ORGANONITRO COMPOUNDS FOR USE IN TREATING NON-HODGKIN'S LYMPHOMA AND LEUKEMIA, AND METHODS RELATING THERETO RADIORX, INC. (US) 2012-06-14 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120149678-A1 Organonitro Compounds for Use in Treating Non-Hodgkin's Lymphoma and Leukemia, and Methods Relating Thereto NPM1, MCL1, BCL9 NEK2 2660/4885SIRT6 1642/4885GAA 1034/4885
US-20140308260-A1 METHODS AND COMPOSITIONS COMPRISING A NITRITE-REDUCTASE PROMOTER FOR TREATMENT OF MEDICAL DISORDERS AND PRESERVATION OF BLOOD PRODUCTS HBB, HBG2, HBZ NEK2 3936/4885SIRT6 1239/4885GAA 2990/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.