SCHEMBL9925601

SCHEMBL9925601

O=Nc1ccc(S)c(N=O)c1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.34
HSD17B10 Q99714 4/20 0.34
TSHR P16473 3/20 0.34
TP53 P04637 2/20 0.34
MAPK1 P28482 2/20 0.34
HIF1A Q16665 2/20 0.34
CYP3A4 P08684 2/20 0.34
TDP1 Q9NUW8 2/20 0.34
MEN1 O00255 1/20 0.34
GMNN O75496 1/20 0.34
LMNA P02545 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2D6 P10635 1/20 0.34
MAPT P10636 1/20 0.34
HPGD P15428 1/20 0.34
ALOX15 P16050 1/20 0.34
CYP2C19 P33261 1/20 0.34
THPO P40225 1/20 0.34
MTOR P42345 1/20 0.34
BLM P54132 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14075868 0.74 ALDH1A1 (0.33) ALDH1A1HSD17B10TSHRTP53MAPK1
SCHEMBL13268128 0.74 ALDH1A1 (0.37) ALDH1A1HSD17B10TSHRTP53MAPK1
SCHEMBL28195239 0.73 ALDH1A1 (0.35) ALDH1A1HSD17B10TSHRTP53MAPK1
SCHEMBL6050007 0.71 CYP3A4 (0.50) ALDH1A1HSD17B10TSHRTP53MAPK1
SCHEMBL12216540 0.71 TDP1 (0.43) ALDH1A1HSD17B10TSHRTP53MAPK1
SCHEMBL12228262 0.71 MAPT (0.40) ALDH1A1HSD17B10TSHRTP53MAPK1
SCHEMBL12693312 0.71 ALDH1A1 (0.34) ALDH1A1HSD17B10TSHRTP53MAPK1
SCHEMBL13329910 0.71 ALDH1A1 (0.34) ALDH1A1HSD17B10TSHRTP53MAPK1
SCHEMBL28246855 0.71 ALDH1A1 (0.34) ALDH1A1HSD17B10TSHRTP53MAPK1
SCHEMBL13901162 0.71 TSHR (0.44) ALDH1A1TSHRTP53MAPK1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120149674-A1 Diaryl Substituted Alkanes MERCK SHARPE & DOHME CORP. (US) 2012-06-14 US disclosed
US-20110003815-A1 DIPHENYL SUBSTITUTED CYCLOALKANES MERCK & CO., INC. 2011-01-06 US disclosed
US-20100222546-A1 METHODS FOR THE PREPARATION OF FUNCTIONALIZED PEPTIDES, PROTEINS AND CARBOHYDRATES AND THEIR CONJUGATES NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2010-09-02 US disclosed
US-20100168076-A1 DIPHENYL SUBSTITUTED ALKANES MERCK SHARP & DOHME CORP. 2010-07-01 US disclosed
US-20100152185-A1 DIPHENYL SUBSTITUTED CYCLOALKANES, COMPOSITIONS CONTAINING SUCH COMPOUNDS AND METHODS OF USE CHU LIN 2010-06-17 US disclosed
US-20090258851-A1 DIARYL SUBSTITUTED ALKANES MERCK SHARP & DOHME CORP. 2009-10-15 US disclosed
US-20080145863-A1 Affinity selected signature peptides for protein identification and quantification PURDUE RESEARCH FOUNDATION (US) 2008-06-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110003815-A1 DIPHENYL SUBSTITUTED CYCLOALKANES PTGIS, PTGS1, LTC4S ALDH1A1 292/4885HSD17B10 508/4885TSHR 4648/4885
US-20100168076-A1 DIPHENYL SUBSTITUTED ALKANES ALOX5, ALOX15, ALOX15B ALDH1A1 173/4885HSD17B10 682/4885TSHR 4425/4885
US-20100152185-A1 DIPHENYL SUBSTITUTED CYCLOALKANES, COMPOSITIONS CONTAINING SUCH COMPOUNDS AND METHODS OF USE ALOX5, LTC4S, ALOX15 ALDH1A1 397/4885HSD17B10 839/4885TSHR 4646/4885
US-20100222546-A1 METHODS FOR THE PREPARATION OF FUNCTIONALIZED PEPTIDES, PROTEINS AND CARBOHYDRATES AND THEIR CONJUGATES PTMS, STT3A, GCG ALDH1A1 3690/4885HSD17B10 2692/4885TSHR 1208/4885
US-20120149674-A1 Diaryl Substituted Alkanes ALOX5, ALOX15, LTB4R2 ALDH1A1 328/4885HSD17B10 655/4885TSHR 4620/4885
US-20090258851-A1 DIARYL SUBSTITUTED ALKANES ALOX5, ALOX15, LTB4R2 ALDH1A1 328/4885HSD17B10 655/4885TSHR 4620/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.