SCHEMBL9925971

SCHEMBL9925971

CC1=C(C#N)C(c2ccc(F)cc2)C2=C(CC(c3cccs3)CC2=O)O1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 14/20 0.45
MAPT P10636 9/20 0.45
HTT P42858 2/20 0.42
CYP3A4 P08684 2/20 0.42
CYP2C9 P11712 2/20 0.42
CYP2C19 P33261 2/20 0.42
MEN1 O00255 5/20 0.39
KMT2A Q03164 5/20 0.39
NPSR1 Q6W5P4 2/20 0.39
CYP1A2 P05177 1/20 0.39
RECQL P46063 1/20 0.39
KDM4E B2RXH2 7/20 0.39
POLB P06746 4/20 0.39
LMNA P02545 4/20 0.39
AGTR1 P30556 1/20 0.39
USP2 O75604 4/20 0.38
HSD17B10 Q99714 4/20 0.38
CASP1 P29466 3/20 0.38
CASP7 P55210 3/20 0.38
TSHR P16473 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9925972 0.82 KDM4E (0.54) ALDH1A1MAPTHTTCYP3A4CYP2C9
SCHEMBL4084506 0.73 ALDH1A1 (0.67) ALDH1A1MAPTHTTMEN1KMT2A
SCHEMBL20988857 0.65 LMNA (0.55) ALDH1A1MAPTHTTCYP3A4CYP2C9
SCHEMBL9925966 0.65 ABCC9 (0.48) ALDH1A1MAPTKMT2ANPSR1KDM4E
SCHEMBL9925969 0.65 KDM4E (0.68) ALDH1A1MAPTNPSR1KDM4EPOLB
SCHEMBL12001639 0.64 KDM4E (0.55) ALDH1A1MAPTHTTMEN1KMT2A
SCHEMBL562770 0.64 ALDH1A1 (0.68) ALDH1A1MAPTHTTCYP3A4CYP2C9
SCHEMBL3129599 0.64 ALDH1A1 (0.72) ALDH1A1MAPTHTTCYP3A4CYP2C9
SCHEMBL6706684 0.63 ALDH1A1 (0.79) ALDH1A1MAPTCYP3A4CYP2C9CYP2C19
SCHEMBL11998882 0.63 KDM4E (0.60) ALDH1A1MAPTHTTCYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012078902-A2 PROTEOSTASIS REGULATORS PROTEOSTASIS THERAPEUTICS, INC. (US) 2012-06-14 WO disclosed