SCHEMBL9939397

SCHEMBL9939397

Nc1ccccc1S(=O)(=O)Nc1cccc(N/C(=N\C(=O)c2ccc(Cl)cc2)NCc2ccc(Cl)cc2F)n1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 3/20 0.40
RXFP1 Q9HBX9 1/20 0.35
ACLY P53396 1/20 0.34
ROCK2 O75116 1/20 0.34
ROCK1 Q13464 1/20 0.34
CCKBR P32239 2/20 0.33
EPHX2 P34913 1/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
MAPT P10636 1/20 0.33
HPGD P15428 1/20 0.33
KMT2A Q03164 1/20 0.33
APOBEC3G Q9HC16 1/20 0.33
CCKAR P32238 2/20 0.33
SCN1A P35498 1/20 0.33
SCN5A Q14524 1/20 0.33
SCN8A Q9UQD0 1/20 0.33
HDAC1 Q13547 3/20 0.33
TRPV1 Q8NER1 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16621983 0.90 IDH1 (0.39) IDH1RXFP1ACLYSCN1ASCN5A
SCHEMBL9939466 0.86 GRM4 (0.38) IDH1RXFP1MEN1KMT2AP2RX7
SCHEMBL9939770 0.86 RXFP1 (0.38) IDH1RXFP1ROCK2ROCK1EPHX2
SCHEMBL16621988 0.84 NAMPT (0.40) ROCK2MEN1ALDH1A1LMNAMAPT
SCHEMBL9938519 0.84 VNN1 (0.37) IDH1RXFP1ROCK2ROCK1TRPV1
SCHEMBL9939437 0.83 RXFP1 (0.39) IDH1RXFP1CCKBRMEN1LMNA
SCHEMBL9939441 0.82 LMNA (0.42) MEN1ALDH1A1LMNAMAPTKMT2A
SCHEMBL9939678 0.82 ROCK2 (0.41) RXFP1ROCK2ROCK1VNN1P2RX7
SCHEMBL9939753 0.81 RXFP1 (0.37) IDH1RXFP1ACLYMEN1LMNA
SCHEMBL9939474 0.79 NAMPT (0.39) IDH1TRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012078869-A1 PYRIDONYL GUANIDINE F1F0-ATPASE INHIBITORS AND THERAPEUTIC USES THEREOF LYCERA CORPORATION (US) 2012-06-14 WO disclosed