SCHEMBL9944833

SCHEMBL9944833

CCNc1cc(NC)c(N)cc1C(=O)NC1CC(F)(F)C1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 2/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
GAA P10253 1/20 0.36
MAPT P10636 1/20 0.36
THRB P10828 1/20 0.36
HPGD P15428 1/20 0.36
HTT P42858 1/20 0.36
GFER P55789 1/20 0.36
PLEC Q15149 1/20 0.36
SPR P35270 1/20 0.34
TYK2 P29597 3/20 0.34
LRRK2 Q5S007 1/20 0.33
ACSS2 Q9NR19 1/20 0.32
ALOX15 P16050 1/20 0.32
HSD17B10 Q99714 1/20 0.32
HTR4 Q13639 1/20 0.31
S100A4 P26447 1/20 0.31
DYRK1A Q13627 1/20 0.31
IRAK4 Q9NWZ3 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9946843 0.88 KDM1A (0.34) KDM1ASPRTYK2LRRK2HSD17B10
SCHEMBL9944832 0.82 HCAR3 (0.40) KDM1AALDH1A1MAPTHTT
SCHEMBL9944733 0.80 RAB9A (0.42) HPGDTYK2S100A4
SCHEMBL9899308 0.77 PTGES (0.46) HPGDTYK2S100A4IRAK4
SCHEMBL9899306 0.77 PTGES (0.46) HPGDTYK2S100A4IRAK4
SCHEMBL9944829 0.75 ALDH1A1 (0.39) KDM4EALDH1A1GAAMAPTHPGD
SCHEMBL9946613 0.73 PTGES (0.46)
SCHEMBL9944890 0.70 CNR2 (0.43) HTR4S100A4
SCHEMBL9946693 0.70 PTGES (0.46) ALDH1A1HPGDHTR4S100A4IRAK4
SCHEMBL9947033 0.70 PTGES (0.46) ALDH1A1HPGDHTR4S100A4IRAK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8674113-B2 Compounds BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-03-18 US disclosed
US-20120149676-A1 NOVEL COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-06-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120149676-A1 NOVEL COMPOUNDS PTGS1, PTGER1, PTGES KDM1A 1720/4885KDM4E 3442/4885ALDH1A1 126/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.