SCHEMBL9947719

SCHEMBL9947719

NC(=O)c1cc(F)cc(C2CCC2)c1

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 3/20 0.42
PARP10 Q53GL7 6/20 0.40
KMO O15229 1/20 0.39
PARP14 Q460N5 3/20 0.37
CES2 O00748 1/20 0.36
CES1 P23141 1/20 0.36
OPRM1 P35372 2/20 0.36
OPRD1 P41143 1/20 0.36
OPRK1 P41145 1/20 0.36
KCNH2 Q12809 1/20 0.36
CYP2C9 P11712 1/20 0.36
GRM5 P41594 1/20 0.35
HDAC1 Q13547 1/20 0.34
HDAC8 Q9BY41 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
PARP15 Q460N3 1/20 0.34
PARP2 Q9UGN5 1/20 0.34
TNKS O95271 1/20 0.34
EPHX1 P07099 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3244198 0.93 PARP1 (0.44) PARP1PARP10KMOPARP14CES2
SCHEMBL30597930 0.93 PARP1 (0.44) PARP1PARP10KMOPARP14CES2
SCHEMBL18284064 0.77 GRIA4 (0.39)
SCHEMBL29615899 0.77 HCAR1 (0.52) KMOCES2CES1
SCHEMBL2407201 0.77 HCAR1 (0.52) KMOCES2CES1
SCHEMBL18878233 0.76 PARP1 (0.48) PARP1PARP2
SCHEMBL7077548 0.74 PARP1 (0.60) PARP1CES2CES1
SCHEMBL259315 0.74 CES2 (0.62) PARP1CES2CES1
SCHEMBL13406258 0.74 ALDH1A1 (0.43) KMOOPRK1CYP2C9HDAC1HDAC8
SCHEMBL17175645 0.74 FAAH (0.59) PARP1PARP10KMOOPRM1OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8207347-B2 Pyridone derivatives as NK3 antagonists H. LUNDBECK A/S (DK) 2012-06-26 US disclosed