SCHEMBL9953313

SCHEMBL9953313

COc1ncc(B2OC(C)(C)C(C)(C)O2)cc1S(=O)(=O)NCC1CC1

nearest known ligand 0.55

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALPL P05186 1/20 0.55
CNR2 P34972 12/20 0.41
CNR1 P21554 6/20 0.41
DGAT1 O75907 1/20 0.37
AAK1 Q2M2I8 1/20 0.36
ALDH1A1 P00352 1/20 0.35
HTT P42858 1/20 0.35
PIK3C3 Q8NEB9 1/20 0.34
NPY5R Q15761 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9952979 0.96 ALPL (0.53) ALPLCNR2CNR1DGAT1AAK1
SCHEMBL23585583 0.95 ALPL (0.51) ALPLCNR2CNR1DGAT1AAK1
SCHEMBL14317989 0.85 ALPL (0.59) ALPLDGAT1AAK1ALDH1A1PIK3C3
SCHEMBL9953535 0.84 ALPL (0.57) ALPLDGAT1AAK1
SCHEMBL9953730 0.84 ALPL (0.57) ALPLDGAT1AAK1ALDH1A1HTT
SCHEMBL9955177 0.83 ALPL (0.56) ALPLDGAT1AAK1ALDH1A1PIK3C3
SCHEMBL9954091 0.82 ALPL (0.61) ALPLDGAT1ALDH1A1
SCHEMBL9953472 0.82 ALPL (0.62) ALPLDGAT1AAK1PIK3C3
SCHEMBL9954766 0.82 ALPL (0.56) ALPLDGAT1ALDH1A1HTTPIK3C3
SCHEMBL9953817 0.82 ALPL (0.56) ALPLALDH1A1HTTPIK3C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012174312-A2 BENZIMIDAZOLE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-12-20 WO disclosed
WO-2012087938-A1 QUINAZOLINONE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-06-28 WO disclosed
WO-2012087938-A1 QUINAZOLINONE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-06-28 WO disclosed
WO-2012037108-A1 AMINOQUINOLINE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-03-22 WO disclosed