SCHEMBL9953556

SCHEMBL9953556

Nc1nc2ccc(I)cc2c(=O)n1-c1ccc(CF)cc1

nearest known ligand 0.43

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CA12 O43570 11/20 0.42
CA1 P00915 11/20 0.42
CA2 P00918 11/20 0.42
CA9 Q16790 11/20 0.42
HCAR1 Q9BXC0 1/20 0.40
PDE4D Q08499 1/20 0.39
POLB P06746 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9954651 0.86 POLB (0.53) CA12CA1CA2CA9POLB
SCHEMBL9955025 0.85 ESR2 (0.41) CA12CA1CA2CA9POLB
SCHEMBL9953324 0.84 HCAR1 (0.50) CA12CA1CA2CA9HCAR1
SCHEMBL9954094 0.83 HCAR1 (0.51) CA12CA1CA2CA9HCAR1
SCHEMBL9954066 0.82 PI4KA (0.46) CA12CA1CA2CA9POLB
SCHEMBL9954423 0.81 POLB (0.41) CA12CA1CA2CA9POLB
SCHEMBL9953024 0.80 CA12 (0.52) CA12CA1CA2CA9
SCHEMBL9954672 0.79 TDO2 (0.52) POLB
SCHEMBL9953800 0.78 POLB (0.41) CA12CA1CA2CA9HCAR1
SCHEMBL9953665 0.78 TGM2 (0.45)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012087938-A1 QUINAZOLINONE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-06-28 WO disclosed