SCHEMBL9956885

SCHEMBL9956885

NC(=O)N1CCC2CNC2C1

nearest known ligand 0.38

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 18/20 0.38
CHRNB4 P30926 18/20 0.38
CHRNA3 P32297 18/20 0.38
CHRNA4 P43681 18/20 0.38
MBTD1 Q05BQ5 1/20 0.34
L3MBTL3 Q96JM7 1/20 0.34
SCN9A Q15858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3579621 0.83 CHRNB2 (0.39) CHRNB2CHRNB4CHRNA3CHRNA4MBTD1
SCHEMBL1586665 0.83 CHRNB2 (0.39) CHRNB2CHRNB4CHRNA3CHRNA4MBTD1
SCHEMBL3580704 0.83 CHRNB2 (0.39) CHRNB2CHRNB4CHRNA3CHRNA4MBTD1
SCHEMBL31453271 0.74 HSD11B1 (0.43) CHRNB2CHRNB4CHRNA3CHRNA4L3MBTL3
SCHEMBL28457915 0.74 MBTD1 (0.38) MBTD1L3MBTL3
SCHEMBL13760961 0.74 GPR119 (0.47)
SCHEMBL928825 0.74 GPR119 (0.47)
SCHEMBL1658442 0.73 KDM4E (0.31)
SCHEMBL4743328 0.73 KDM1A (0.37) MBTD1L3MBTL3
SCHEMBL3332672 0.72 CHRNB2 (0.56) CHRNB2CHRNB4CHRNA3CHRNA4MBTD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012085857-A1 3,8-DIAZA-BICYCLO[4.2.0]OCT-3-YL AMIDES ACTELION PHARMACEUTICALS LTD (CH) 2012-06-28 WO disclosed
WO-2012085857-A1 3,8-DIAZA-BICYCLO[4.2.0]OCT-3-YL AMIDES ACTELION PHARMACEUTICALS LTD (CH) 2012-06-28 WO disclosed