SCHEMBL9957060

SCHEMBL9957060

c1ccc(C(=Nc2cccnn2)c2ccccc2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TBXA2R P21731 1/20 0.40
ESR1 P03372 1/20 0.37
ESR2 Q92731 1/20 0.37
VNN1 O95497 1/20 0.34
ADRA2A P08913 2/20 0.33
ADRA2B P18089 2/20 0.33
ADRA2C P18825 2/20 0.33
PLAU P00749 1/20 0.33
GAA P10253 1/20 0.33
SMN1; SMN2 Q16637 3/20 0.32
ALDH1A1 P00352 2/20 0.32
CYP1A2 P05177 2/20 0.32
BCHE P06276 1/20 0.32
AGTR1 P30556 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
HPGD P15428 1/20 0.32
CYP2C19 P33261 1/20 0.32
MEN1 O00255 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2729935 0.76 ADRA2A (0.59) ADRA2AADRA2BADRA2CPLAUGAA
SCHEMBL31465345 0.73 ALDH1A1 (0.38) ESR1ESR2GAASMN1; SMN2ALDH1A1
SCHEMBL28294254 0.72 TBXA2R (0.42) TBXA2RESR1ESR2ADRA2AADRA2B
SCHEMBL2013760 0.72 TBXA2R (0.52) TBXA2RVNN1GAASMN1; SMN2ALDH1A1
SCHEMBL2013758 0.72 TBXA2R (0.52) TBXA2RVNN1GAASMN1; SMN2ALDH1A1
SCHEMBL30189924 0.72 TBXA2R (0.42) TBXA2RESR1ESR2ADRA2AADRA2B
SCHEMBL30281198 0.72 GFER (0.36) ESR1ESR2PLAUSMN1; SMN2KMT2A
SCHEMBL9950334 0.72 GFER (0.36) ESR1ESR2PLAUSMN1; SMN2KMT2A
SCHEMBL1853792 0.69 MAOA (0.41) ALDH1A1CYP1A2GOT1DHODH
SCHEMBL27983624 0.69 GOT1 (0.41) CYP1A2GOT1P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116390917-A MRGX2 antagonists 葛兰素史密斯克莱知识产权发展有限公司 2023-07-04 CN disclosed
WO-2012088266-A2 SUBSTITUTED IMIDAZOPYRIDAZINES AND BENZIMIDAZOLES AS INHIBITORS OF FGFR3 INCYTE CORPORATION (US) 2012-06-28 WO disclosed