SCHEMBL998674

SCHEMBL998674

COC(=O)C(C)c1[c]cccc1

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.43
PTGS1 P23219 1/20 0.43
PTGS2 P35354 1/20 0.43
HPGD P15428 2/20 0.37
MAPT P10636 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
MEN1 O00255 2/20 0.36
KDM1A O60341 1/20 0.36
ALDH1A1 P00352 2/20 0.35
KDM4E B2RXH2 1/20 0.35
TSHR P16473 1/20 0.34
MT-CO2 P00403 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4816673 0.83 TSHR (0.43) KMT2AHPGDMAPTL3MBTL1MEN1
SCHEMBL11285004 0.81 L3MBTL1 (0.44) KMT2APTGS1HPGDMAPTL3MBTL1
SCHEMBL11276127 0.81 GAA (0.41) HPGDMAPTL3MBTL1ALDH1A1
SCHEMBL27447903 0.81 KMT2A (0.42) KMT2AMEN1ALDH1A1TSHR
SCHEMBL4016238 0.79 PTGS2 (0.46) KMT2APTGS1PTGS2HPGDMAPT
SCHEMBL11286164 0.79 ALDH1A1 (0.49) KMT2AL3MBTL1ALDH1A1
SCHEMBL3539841 0.78 KMT2A (0.40) KMT2AMAPTL3MBTL1MEN1ALDH1A1
SCHEMBL11043246 0.78 EPHX1 (0.37) KMT2APTGS2MAPTL3MBTL1KDM1A
SCHEMBL11409716 0.77 NLRP3 (0.45) KMT2AMEN1ALDH1A1KDM4ETSHR
SCHEMBL11281869 0.77 LMNA (0.40) KMT2AHPGDMAPTL3MBTL1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2456435-A1 HETEROARYL BENZAMIDES, COMPOSITIONS AND METHODS OF USE The Board of Trustees of The Leland Stanford Junior University (US) 2012-05-30 EP disclosed
WO-2011011514-A1 HETEROARYL BENZAMIDES, COMPOSITIONS AND METHODS OF USE THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2011-01-27 WO disclosed