SCHEMBL9987009

SCHEMBL9987009

O=C(O)C1CCN(c2ccc(Nc3nc(NCCCn4ccnc4)ccc3[N+](=O)[O-])cc2F)CC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 3/20 0.46
ALDH1A1 P00352 3/20 0.46
KMT2A Q03164 3/20 0.46
MAPT P10636 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
MEN1 O00255 2/20 0.46
MAPK1 P28482 1/20 0.45
HTT P42858 1/20 0.45
TDP1 Q9NUW8 1/20 0.39
CYP19A1 P11511 1/20 0.39
SERPINE1 P05121 1/20 0.38
EGFR P00533 1/20 0.38
MAOA P21397 1/20 0.36
MAOB P27338 1/20 0.36
QPCT Q16769 1/20 0.36
JAK2 O60674 1/20 0.36
BRD4 O60885 1/20 0.36
NAMPT P43490 3/20 0.35
RET P07949 1/20 0.35
ROS1 P08922 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9984101 0.94 ALDH1A1 (0.45) L3MBTL1ALDH1A1KMT2AMAPTSMN1; SMN2
SCHEMBL9984090 0.87 ALDH1A1 (0.45) L3MBTL1ALDH1A1KMT2AMAPTSMN1; SMN2
SCHEMBL9987164 0.84 TDP1 (0.42) L3MBTL1ALDH1A1KMT2AMAPTSMN1; SMN2
SCHEMBL9983509 0.83 ALDH1A1 (0.42) L3MBTL1ALDH1A1KMT2AMAPTSMN1; SMN2
SCHEMBL9987060 0.82 TDP1 (0.43) KMT2AMAPTMEN1MAPK1TDP1
SCHEMBL9987376 0.81 TDP1 (0.48) L3MBTL1KMT2AMAPTMEN1MAPK1
SCHEMBL9987013 0.81 TDP1 (0.39) TDP1SERPINE1JAK2BRD4RET
SCHEMBL9987425 0.81 MAPT (0.44) ALDH1A1MAPTHTTTDP1SERPINE1
SCHEMBL9987584 0.79 BRD4 (0.51) L3MBTL1KMT2AMAPTMEN1MAPK1
SCHEMBL9987980 0.78 TDP1 (0.49) L3MBTL1KMT2AMAPTMEN1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2394993-A2 NOVEL 2,6-SUBSTITUTED-3-NITROPYRIDINE DERIVATIVE, METHOD FOR PREPARING SAME, AND PHARMACEUTICAL COMPOSITION INCLUDING SAME Dong Wha Pharm. Co., Ltd. (KR) 2011-12-14 EP disclosed