SCHEMBL10018709

SCHEMBL10018709

Cc1cc(F)c(-c2ccc(C)c(F)c2)c(F)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NISCH Q9Y2I1 1/20 0.47
AKR1C3 P42330 2/20 0.41
AKR1C2 P52895 2/20 0.41
HDAC1 Q13547 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
KMO O15229 2/20 0.39
ERN1 O75460 1/20 0.37
ESR1 P03372 1/20 0.37
ESR2 Q92731 1/20 0.37
PDE3B Q13370 1/20 0.37
PDE3A Q14432 1/20 0.37
AKR1B10 O60218 1/20 0.36
AKR1C4 P17516 1/20 0.36
AKR1C1 Q04828 1/20 0.36
DHODH Q02127 2/20 0.36
ACHE P22303 1/20 0.36
SLC6A3 Q01959 1/20 0.36
BRD4 O60885 1/20 0.35
CREBBP Q92793 1/20 0.35
PTGS2 P35354 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22219382 0.89 NISCH (0.42) NISCHAKR1C3AKR1C2HDAC1HDAC6
SCHEMBL14365641 0.88 NISCH (0.45) NISCHAKR1C3AKR1C2KMOERN1
SCHEMBL13087002 0.87 NISCH (0.43) NISCHAKR1C3AKR1C2HDAC1HDAC6
SCHEMBL17407511 0.83 ESR1 (0.56) NISCHAKR1C3AKR1C2HDAC1HDAC6
SCHEMBL10014272 0.83 NFE2L2 (0.48) AKR1C3AKR1C2ESR1ESR2DHODH
SCHEMBL24540157 0.82 AKR1C3 (0.38) NISCHAKR1C3AKR1C2HDAC1HDAC6
SCHEMBL19807356 0.82 PTGS2 (0.48) KMODHODHPTGS2PTGS1
SCHEMBL12377626 0.81 NISCH (0.52) NISCHAKR1C3AKR1C2HDAC1HDAC6
SCHEMBL91695 0.80 ERN1 (0.47) NISCHAKR1C3AKR1C2KMOERN1
SCHEMBL10304803 0.80 NISCH (0.44) NISCHAKR1C3AKR1C2HDAC1HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 66 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11834599-B2 Aromatic isothiocyanates MERCK PATENT GMBH (DE) 2023-12-05 US disclosed
US-11739265-B2 Aromatic isothiocyanates MERCK PATENT GMBH (DE) 2023-08-29 US disclosed
US-11667841-B2 Dibenzofuran and dibenzothiophene derivatives MERCK PATENT GMBH (DE) 2023-06-06 US disclosed
US-11312908-B2 Liquid crystal medium and liquid crystal display MERCK PATENT GMBH (DE) 2022-04-26 US disclosed
US-11268026-B2 Liquid-crystalline medium MERCK PATENT GMBH (DE) 2022-03-08 US disclosed
US-20210403810-A1 DIBENZOFURAN AND DIBENZOTHIOPHENE DERIVATIVES MERCK PATENT GMBH (DE) 2021-12-30 US disclosed
US-11208594-B2 Liquid-crystalline medium and high-frequency components comprising same MERCK PATENT GMBH (DE) 2021-12-28 US disclosed
US-20210115337-A1 LIQUID-CRYSTALLINE MEDIUM MERCK PATENT GMBH (DE) 2021-04-22 US disclosed
US-20210102122-A1 LIQUID CRYSTAL MEDIUM MERCK PATENT GMBH (DE) 2021-04-08 US disclosed
US-10711197-B2 Liquid-crystalline medium and high-frequency components comprising same MERCK PATENT GMBH (DE) 2020-07-14 US disclosed
EP-1816180-B1 Mesogenic compounds, liquid crystal medium, and liquid crystal display MERCK PATENT GMBH (DE) 2008-10-29 EP disclosed
EP-1690917-B1 Mesogenic compounds, liquid crystal medium and liquid crystal display MERCK PATENT GMBH (DE) 2008-10-08 EP disclosed
US-20080167482-A1 mesogenic group is linked to the C-atom No. 5 of the 1,3-dioxane-5-yl group; media showing a blue phase and their use in electro-optical light modulation elements MERCK PATENT GMBH (DE) 2008-07-10 US disclosed
US-20080167482-A1 mesogenic group is linked to the C-atom No. 5 of the 1,3-dioxane-5-yl group; media showing a blue phase and their use in electro-optical light modulation elements MERCK PATENT GMBH (DE) 2008-07-10 US disclosed
US-20080116419-A1 Mesogenic Compounds, Liquid Crystal Medium and Liquid Crystal Display MERCK PATENT GMBH (DE) 2008-05-22 US disclosed
US-20080116419-A1 Mesogenic Compounds, Liquid Crystal Medium and Liquid Crystal Display MERCK PATENT GMBH (DE) 2008-05-22 US disclosed
EP-1690915-B1 Mesogenic compounds, liquid crystal medium and liquid crystal display MERCK PATENT GMBH (DE) 2008-03-26 EP disclosed
EP-1690916-B1 Mesogenic compounds, liquid crystal medium and liquid crystal display MERCK PATENT GMBH (DE) 2008-03-12 EP disclosed
EP-1816180-A1 Mesogenic compounds, liquid crystal medium, and liquid crystal display Merck Patent GmbH (DE) 2007-08-08 EP disclosed
EP-1739151-A1 Mesogenic compounds, liquid crystal medium and liquid display MERCK PATENT GmbH (DE) 2007-01-03 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11667841-B2 Dibenzofuran and dibenzothiophene derivatives DDT, MYT1, DBF4 NISCH 196/4885AKR1C3 4097/4885AKR1C2 4331/4885
US-20210403810-A1 DIBENZOFURAN AND DIBENZOTHIOPHENE DERIVATIVES DDT, MYT1, DBF4 NISCH 196/4885AKR1C3 4097/4885AKR1C2 4331/4885
US-20080116419-A1 Mesogenic Compounds, Liquid Crystal Medium and Liquid Crystal Display CRY1, CRY2, IK NISCH 126/4885AKR1C3 2896/4885AKR1C2 3229/4885
US-11739265-B2 Aromatic isothiocyanates TRPA1, CRY1, FOXM1 NISCH 202/4885AKR1C3 3786/4885AKR1C2 3646/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.