SCHEMBL1003443

SCHEMBL1003443

COC(=O)c1cc(C(O)(CC(=O)OC(C)(C)C)Cc2ccc(Br)cc2)cn1C(=O)O

nearest known ligand 0.33

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.33
CTSS P25774 1/20 0.32
CTSK P43235 1/20 0.32
LMNA P02545 1/20 0.32
GAA P10253 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30
ALDH1A1 P00352 2/20 0.30
KDM4E B2RXH2 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2C9 P11712 1/20 0.30
HPGD P15428 1/20 0.30
CYP2C19 P33261 1/20 0.30
MAPK10 P53779 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2075856 0.92 PTGS2 (0.33) PTGS2CTSSCTSKLMNAGAA
SCHEMBL1003620 0.71 ALDH1A1 (0.41) PTGS2LMNAGAANPSR1L3MBTL1
SCHEMBL2076144 0.69 HDAC1 (0.36) PTGS2CTSSCTSKLMNAGAA
SCHEMBL20141700 0.66 KDM4E (0.36) GAANPSR1L3MBTL1ALDH1A1KDM4E
SCHEMBL4131647 0.63 NR1H2 (0.42) LMNAL3MBTL1KDM4E
SCHEMBL4610689 0.63 FPR2 (0.38) LMNAGAAALDH1A1KDM4E
SCHEMBL5533824 0.62 MTNR1A (0.46) CTSSCTSKLMNAL3MBTL1ALDH1A1
SCHEMBL15270503 0.60 CACNA1B (0.42) CTSSCTSKLMNAALDH1A1KDM4E
SCHEMBL31048202 0.60 L3MBTL1 (0.44) CTSSCTSKLMNAL3MBTL1ALDH1A1
SCHEMBL28797147 0.60 SMN1; SMN2 (0.43) CTSSCTSKLMNAL3MBTL1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011011330-A2 INHIBITORS OF D-AMINO ACID OXIDASE SEPRACOR INC. (US) 2011-01-27 WO disclosed