SCHEMBL1011331

SCHEMBL1011331

N#Cc1cccc2c1CCNC2CI

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.40
GID4 Q8IVV7 2/20 0.37
PRCP P42785 2/20 0.35
SLC22A1 O15245 1/20 0.35
HTR2C P28335 1/20 0.35
HTR2B P41595 1/20 0.35
KDM1A O60341 1/20 0.34
S1PR1 P21453 2/20 0.34
S1PR3 Q99500 1/20 0.34
SLC6A4 P31645 2/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A3 Q01959 1/20 0.33
PNMT P11086 1/20 0.33
DRD1 P21728 1/20 0.32
DRD4 P21917 1/20 0.32
DRD5 P21918 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1487596 0.76 PDE9A (0.38) DRD2GID4HTR2CHTR2BKDM1A
SCHEMBL4019842 0.71 ADRA2A (0.46)
SCHEMBL4020963 0.70 PRCP (0.65) PRCPSLC22A1
SCHEMBL4020702 0.70 PRCP (0.65) PRCPSLC22A1
SCHEMBL1009372 0.69 OPRK1 (0.36) GID4PRCPSLC22A1S1PR1S1PR3
SCHEMBL33532651 0.66 GID4 (0.52) DRD2GID4PRCPSLC22A1HTR2C
SCHEMBL33531851 0.66 GID4 (0.56) GID4PRCPSLC22A1HTR2CHTR2B
SCHEMBL25193256 0.64 DRD2 (0.45) DRD2HTR2CHTR2BS1PR1SLC6A4
SCHEMBL12420776 0.64 DRD2 (0.45) DRD2S1PR1S1PR3DRD1DRD4
SCHEMBL2196969 0.64 KMT2A (0.50) DRD2S1PR1DRD1DRD4DRD5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2054416-B1 SUBSTITUTED PYRAZOLOPYRIMIDINES, A PROCESS FOR THEIR PREPARATION AND THEIR USE AS MEDICINE MERZ PHARMA GMBH & CO KGAA (DE) 2011-01-05 EP disclosed