SCHEMBL10122342

SCHEMBL10122342

c1ccc(-c2c3ccccc3c(-c3c4oc5ccccc5c4cc4c3oc3ccccc34)c3ccccc23)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AHR P35869 3/20 0.46
CA1 P00915 3/20 0.44
CA2 P00918 3/20 0.44
HPGD P15428 4/20 0.42
CYP3A4 P08684 3/20 0.42
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
CA12 O43570 2/20 0.42
TP53 P04637 2/20 0.42
ABCB1 P08183 2/20 0.42
ADORA3 P0DMS8 2/20 0.42
AR P10275 2/20 0.42
CYP1B1 Q16678 2/20 0.42
CA9 Q16790 2/20 0.42
GABRP O00591 1/20 0.42
GABRD O14764 1/20 0.42
TNKS O95271 1/20 0.42
PARP1 P09874 1/20 0.42
CYP19A1 P11511 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10122330 0.97 AHR (0.44) AHRCA1CA2HPGDCYP3A4
SCHEMBL10122352 0.93 AHR (0.46) AHRCA1CA2HPGDCYP3A4
SCHEMBL10122344 0.91 AHR (0.45) AHRCA1CA2HPGDCYP3A4
SCHEMBL10122693 0.91 AHR (0.53) AHRCA1HPGDCYP3A4NPC1
SCHEMBL10122335 0.90 PLA2G2A (0.43) AHRCA1CA2HPGDCYP3A4
SCHEMBL10122366 0.90 AHR (0.44) AHRCA1CA2HPGDCYP3A4
SCHEMBL17932160 0.88 AHR (0.42) AHRCA1CA2HPGDCYP3A4
SCHEMBL19081432 0.87 ABCG2 (0.45) AHRCA1CA2HPGDCYP3A4
SCHEMBL10122624 0.87 AHR (0.41) AHRCA1CA2HPGDCYP3A4
SCHEMBL10122363 0.87 PLA2G2A (0.43) AHRCA1CA2HPGDCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 47 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12030900-B2 Boron compound and organic light-emitting diode comprising same SFC CO., LTD. (KR) 2024-07-09 US disclosed
US-12018039-B2 Boron compound, and organic light-emitting diode comprising same SFC CO., LTD. (KR) 2024-06-25 US disclosed
US-20240018164-A1 POLYCYCLIC AROMATIC DERIVATIVE COMPOUND AND ORGANOELECTROLUMINESCENT DEVICE USING SAME SFC CO., LTD. (KR) 2024-01-18 US disclosed
US-20230371376-A1 POLYCYCLIC COMPOUND AND ORGANIC LIGHT-EMITTING DEVICE USING SAME SFC CO., LTD. (KR) 2023-11-16 US disclosed
US-20230329025-A1 ORGANIC ELECTROLUMINESCENT ELEMENT AND ELECTRONIC DEVICE IDEMITSU KOSAN CO.,LTD. (JP) 2023-10-12 US disclosed
US-20230329109-A1 POLYCYCLIC AROMATIC DERIVATIVE COMPOUND AND ORGANOELECTROLUMINESCENT DEVICE USING SAME SFC CO., LTD. (KR) 2023-10-12 US disclosed
US-20230329025-A1 ORGANIC ELECTROLUMINESCENT ELEMENT AND ELECTRONIC DEVICE IDEMITSU KOSAN CO.,LTD. (JP) 2023-10-12 US disclosed
US-20230287010-A1 POLYCYCLIC AROMATIC DERIVATIVE COMPOUND AND ORGANIC LIGHT-EMITTING DEVICE USING SAME SFC CO., LTD (KR) 2023-09-14 US disclosed
US-20230284515-A1 POLYCYCLIC AROMATIC DERIVATIVE COMPOUND AND ORGANIC LIGHT-EMITTING ELEMENT USING THE SAME SFC CO., LTD. (KR) 2023-09-07 US disclosed
US-20230189646-A1 POLYCYCLIC AROMATIC COMPOUND AND ORGANOELECTROLUMINESCENT DEVICE USING SAME SFC CO., LTD (KR) 2023-06-15 US disclosed
US-20140159005-A1 ANTHRACENE DERIVATIVE AND ORGANIC ELECTROLUMINESCENT ELEMENT USING THE SAME IIDEMITSU KOSAN CO., LTD (JP) 2014-06-12 US disclosed
US-20140061622-A1 ORGANIC ELECTROLUMINESCENCE DEVICE IDEMITSU KOSAN CO., LTD. (JP) 2014-03-06 US disclosed
EP-2700696-A1 PYRENE DERIVATIVE, ORGANIC LIGHT-EMITTING MEDIUM, AND ORGANIC ELECTROLUMINESCENT ELEMENT CONTAINING PYRENE DERIVATIVE OR ORGANIC LIGHT-EMITTING MEDIUM Idemitsu Kosan Co., Ltd (JP) 2014-02-26 EP disclosed
US-20140034943-A1 PYRENE DERIVATIVE, ORGANIC LIGHT-EMITTING MEDIUM, AND ORGANIC ELECTROLUMINESCENT ELEMENT CONTAINING PYRENE DERIVATIVE OR ORGANIC LIGHT-EMITTING MEDIUM IDEMITSU KOSAN CO., LTD. 2014-02-06 US disclosed
US-20140034943-A1 PYRENE DERIVATIVE, ORGANIC LIGHT-EMITTING MEDIUM, AND ORGANIC ELECTROLUMINESCENT ELEMENT CONTAINING PYRENE DERIVATIVE OR ORGANIC LIGHT-EMITTING MEDIUM IDEMITSU KOSAN CO., LTD. 2014-02-06 US disclosed
US-8629430-B2 Anthracene derivative and organic electroluminescent element using the same IDEMITSU KOSAN CO., LTD. (JP) 2014-01-14 US disclosed
US-8629430-B2 Anthracene derivative and organic electroluminescent element using the same IDEMITSU KOSAN CO., LTD. (JP) 2014-01-14 US disclosed
US-20120138914-A1 ANTHRACENE DERIVATIVE AND ORGANIC ELECTROLUMINESCENT ELEMENT USING THE SAME IDEMITSU KOSAN CO., LTD. (JP) 2012-06-07 US disclosed
US-20120138914-A1 ANTHRACENE DERIVATIVE AND ORGANIC ELECTROLUMINESCENT ELEMENT USING THE SAME IDEMITSU KOSAN CO., LTD. (JP) 2012-06-07 US disclosed
WO-2010137285-A1 ANTHRACENE DERIVATIVE AND ORGANIC ELECTROLUMINESCENT ELEMENT USING THE SAME 出光興産株式会社 (JP) 2010-12-02 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (10 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230287010-A1 POLYCYCLIC AROMATIC DERIVATIVE COMPOUND AND ORGANIC LIGHT-EMITTING DEVICE USING SAME DDT, TYR, DDC AHR 19/4885CA1 4833/4885CA2 4746/4885
US-20140159005-A1 ANTHRACENE DERIVATIVE AND ORGANIC ELECTROLUMINESCENT ELEMENT USING THE SAME SOX18, ANXA1, ANXA11 AHR 314/4885CA1 230/4885CA2 547/4885
US-12018039-B2 Boron compound, and organic light-emitting diode comprising same CLTB, CD79B, CYBA AHR 491/4885CA1 3149/4885CA2 1600/4885
US-20230371376-A1 POLYCYCLIC COMPOUND AND ORGANIC LIGHT-EMITTING DEVICE USING SAME PPOX, MAP1LC3A, VDAC2 AHR 64/4885CA1 3702/4885CA2 3947/4885
US-20120138914-A1 ANTHRACENE DERIVATIVE AND ORGANIC ELECTROLUMINESCENT ELEMENT USING THE SAME SOX18, ANXA1, ANXA11 AHR 314/4885CA1 230/4885CA2 547/4885
US-20240018164-A1 POLYCYCLIC AROMATIC DERIVATIVE COMPOUND AND ORGANOELECTROLUMINESCENT DEVICE USING SAME DDT, UROD, DDC AHR 12/4885CA1 4783/4885CA2 4090/4885
US-20230284515-A1 POLYCYCLIC AROMATIC DERIVATIVE COMPOUND AND ORGANIC LIGHT-EMITTING ELEMENT USING THE SAME ARNT, AHR, TYR AHR 2/4885CA1 2614/4885CA2 2631/4885
US-20230329109-A1 POLYCYCLIC AROMATIC DERIVATIVE COMPOUND AND ORGANOELECTROLUMINESCENT DEVICE USING SAME DDT, UROD, DDC AHR 14/4885CA1 4794/4885CA2 4282/4885
US-20230189646-A1 POLYCYCLIC AROMATIC COMPOUND AND ORGANOELECTROLUMINESCENT DEVICE USING SAME DDC, DDT, AHR AHR 3/4885CA1 4796/4885CA2 4718/4885
US-12030900-B2 Boron compound and organic light-emitting diode comprising same CLTB, CD79B, CYBA AHR 656/4885CA1 3133/4885CA2 1404/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.