Cycloproparadicicol

Cycloproparadicicol

SCHEMBL10149963

C[C@@H]1C[C@H]2C[C@@H]2/C=C\C=C\C(=O)Cc2c(Cl)c(O)cc(O)c2C(=O)O1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AB1 P08238 4/20 1.00
MAPT P10636 3/20 0.73
HSP90AA1 P07900 2/20 0.73
GAA P10253 1/20 0.73
RAB9A P51151 1/20 0.73
NPSR1 Q6W5P4 1/20 0.73
NLRP3 Q96P20 1/20 0.73
CBR1 P16152 1/20 0.73
PTGS2 P35354 1/20 0.73
ACLY P53396 1/20 0.73
FTO Q9C0B1 1/20 0.73
MEN1 O00255 1/20 0.73
ALDH1A1 P00352 1/20 0.73
HPGD P15428 1/20 0.73
KMT2A Q03164 1/20 0.73
KDM4E B2RXH2 1/20 0.42
POLB P06746 1/20 0.42
STAT6 P42226 1/20 0.39
SMAD3 P84022 1/20 0.39
SMAD2 Q15796 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Cycloproparadicicol SCHEMBL20840799 1.00 HSP90AB1 (1.00) HSP90AB1MAPTHSP90AA1GAARAB9A
Cycloproparadicicol SCHEMBL10150412 1.00 HSP90AB1 (1.00) HSP90AB1MAPTHSP90AA1GAARAB9A
Cycloproparadicicol SCHEMBL14212855 1.00 HSP90AB1 (1.00) HSP90AB1MAPTHSP90AA1GAARAB9A
Cycloproparadicicol SCHEMBL2622302 1.00 HSP90AB1 (1.00) HSP90AB1MAPTHSP90AA1GAARAB9A
SCHEMBL19418326 0.92 HSP90AB1 (0.85) HSP90AB1MAPTHSP90AA1GAARAB9A
SCHEMBL14212857 0.89 HSP90AB1 (0.80) HSP90AB1MAPTHSP90AA1GAARAB9A
SCHEMBL14212864 0.89 HSP90AB1 (0.80) HSP90AB1MAPTHSP90AA1GAARAB9A
SCHEMBL14182170 0.89 HSP90AB1 (0.80) HSP90AB1MAPTHSP90AA1GAARAB9A
SCHEMBL14182165 0.89 HSP90AB1 (0.80) HSP90AB1MAPTHSP90AA1GAARAB9A
SCHEMBL10149964 0.89 HSP90AB1 (0.80) HSP90AB1MAPTHSP90AA1GAARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 34 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3782649-B1 BIODEGRADABLE POLYETHYLENE GLYCOL BASED WATER-INSOLUBLE HYDROGELS ASCENDIS PHARMA AS (DK) 2025-05-14 EP disclosed
US-11873310-B2 Compounds useful in HIV therapy GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2024-01-16 US disclosed
US-20230381323-A1 RELEASABLE CONJUGATES FISH & RICHARDSON PC 2023-11-30 US disclosed
US-11786599-B2 Releasable conjugates QUIAPEG PHARMACEUTICALS AB (SE) 2023-10-17 US disclosed
US-20230123784-A1 Biodegradable Polyethylene Glycol Based Water-Insoluble Hydrogels ASCENDIS PHARMA A/S (DK) 2023-04-20 US disclosed
US-11559482-B2 Biodegradable polyethylene glycol based water-insoluble hydrogels ASCENDIS PHARMA A/S (DE) 2023-01-24 US disclosed
EP-4011396-A1 RELEASABLE CONJUGATES QuiaPEG Pharmaceuticals AB (SE) 2022-06-15 EP disclosed
US-20220119417-A1 Compounds Useful in HIV Therapy GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2022-04-21 US disclosed
US-10975056-B2 Substituted pyridines as inhibitors of DNMT1 GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2021-04-13 US disclosed
US-20210009609-A1 Compounds Useful in HIV Therapy GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2021-01-14 US disclosed
US-20120077775-A1 MACROCYCLIC COMPOUNDS USEFUL AS INHIBITORS OF KINASES AND HSP90 LE CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2012-03-29 US disclosed
US-8067412-B2 analogs of natural products radicicol and pochonins; (oxirane or cyclopropan) 2-benzoxacyclo(di)tetradecin derivatives; inhibition of kinase phosphorylation activity and heat shock proteins; anticarcinogenic, antiinflammatory agent; neurodegenerative diseases; antiallergen UNIVERSITE DE STRASBOURG (FR) 2011-11-29 US disclosed
US-20110190237-A1 Macrocyclic Prodrug Compounds Useful as Therapeutics NEXGENIX PHARMACEUTICALS (US) 2011-08-04 US disclosed
US-20100292218-A1 Treatment Of Neurofibromatosis With Radicicol And Its Derivatives NEXGENIX PHARMACEUTICALS HOLDINGS, INC. 2010-11-18 US disclosed
US-20100093824-A1 METHODS OF TREATING VIRAL INFECTION THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2010-04-15 US disclosed
US-20100093824-A1 METHODS OF TREATING VIRAL INFECTION THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2010-04-15 US disclosed
WO-2008143647-A2 METHODS OF TREATING VIRAL INFECTION THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2008-11-27 WO disclosed
US-20080146545-A1 Macrocyclic compounds useful as inhibitors of kinases and HSP90 UNIVERSITE DE STRASBOURG (FR) 2008-06-19 US disclosed
US-20080108694-A1 Novel Macrocycles and Uses Thereof NATIONAL INSTITUTES OF HEALTH - DIRECTOR DEITR 2008-05-08 US disclosed
US-20080108694-A1 Novel Macrocycles and Uses Thereof NATIONAL INSTITUTES OF HEALTH - DIRECTOR DEITR 2008-05-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (14 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080108694-A1 Novel Macrocycles and Uses Thereof BDKRB1, RPS4Y1, GRK4 HSP90AB1 3784/4885MAPT 4737/4885HSP90AA1 4330/4885
US-20120077775-A1 MACROCYCLIC COMPOUNDS USEFUL AS INHIBITORS OF KINASES AND HSP90 HSP90AB1, HSP90AA1, HSP90AB2P HSP90AB1 1/4885MAPT 1982/4885HSP90AA1 2/4885
US-20220119417-A1 Compounds Useful in HIV Therapy CD4, CCR5, ABCB1 HSP90AB1 1471/4885MAPT 650/4885HSP90AA1 2339/4885
US-20100093824-A1 METHODS OF TREATING VIRAL INFECTION EIF2AK2, NSUN2, NSUN3 HSP90AB1 250/4885MAPT 2183/4885HSP90AA1 375/4885
US-11873310-B2 Compounds useful in HIV therapy CD4, CCR5, ABCB1 HSP90AB1 1471/4885MAPT 650/4885HSP90AA1 2339/4885
US-20100292218-A1 Treatment Of Neurofibromatosis With Radicicol And Its Derivatives HSP90AB2P, HSP90AA1, HSPA2 HSP90AB1 4/4885MAPT 2339/4885HSP90AA1 2/4885
US-20230123784-A1 Biodegradable Polyethylene Glycol Based Water-Insoluble Hydrogels PLG, PHYKPL, PLOD3 HSP90AB1 80/4885MAPT 1671/4885HSP90AA1 164/4885
US-10975056-B2 Substituted pyridines as inhibitors of DNMT1 DNMT1, DNMT3A, DNMT3B HSP90AB1 4339/4885MAPT 3289/4885HSP90AA1 4617/4885
US-20230381323-A1 RELEASABLE CONJUGATES GUSB, ABCB11, UGT2B7 HSP90AB1 320/4885MAPT 3354/4885HSP90AA1 984/4885
US-20080146545-A1 Macrocyclic compounds useful as inhibitors of kinases and HSP90 HSP90AB1, HSP90AA1, HSP90AB2P HSP90AB1 1/4885MAPT 1982/4885HSP90AA1 2/4885
US-20110190237-A1 Macrocyclic Prodrug Compounds Useful as Therapeutics ADCYAP1R1, CYP19A1, THOP1 HSP90AB1 3953/4885MAPT 2173/4885HSP90AA1 4055/4885
US-11559482-B2 Biodegradable polyethylene glycol based water-insoluble hydrogels PLG, PHYKPL, PLOD3 HSP90AB1 80/4885MAPT 1671/4885HSP90AA1 164/4885
US-11786599-B2 Releasable conjugates GUSB, ABCB11, UGT2B7 HSP90AB1 320/4885MAPT 3354/4885HSP90AA1 984/4885
US-20210009609-A1 Compounds Useful in HIV Therapy CD4, CCR5, ABCB1 HSP90AB1 2177/4885MAPT 876/4885HSP90AA1 2660/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.