SCHEMBL10153995

SCHEMBL10153995

COC(=O)C1C(=O)N(OCc2ccccc2)C(=O)c2cc(NC(=O)c3ccccn3)ccc21

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GRM4 Q14833 11/20 0.44
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
KDM4E B2RXH2 1/20 0.44
KDR P35968 2/20 0.43
HDAC6 Q9UBN7 1/20 0.42
FTO Q9C0B1 1/20 0.42
MAPT P10636 1/20 0.41
PKM P14618 1/20 0.41
KCNK3 O14649 1/20 0.41
KCNK9 Q9NPC2 1/20 0.41
GRM1 Q13255 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10153293 0.88 ACHE (0.45) NPC1RAB9ASMN1; SMN2MAPTKCNK9
SCHEMBL10153594 0.86 ACHE (0.45) NPC1RAB9ASMN1; SMN2KDM4EMAPT
SCHEMBL10153721 0.84 KDR (0.47) GRM4KDRMAPT
SCHEMBL9959325 0.83 APP (0.42) MAPT
SCHEMBL10153305 0.83 MEN1 (0.46) NPC1RAB9ASMN1; SMN2MAPT
SCHEMBL10153644 0.79 ALDH1A1 (0.42) NPC1RAB9ASMN1; SMN2MAPT
SCHEMBL9959247 0.79 ALDH1A1 (0.42) SMN1; SMN2KDM4EMAPT
SCHEMBL10153698 0.79 ALDH1A1 (0.39) KDM4EMAPT
SCHEMBL9960564 0.79 TRPA1 (0.38) MAPT
SCHEMBL10153686 0.79 MEN1 (0.46) NPC1RAB9ASMN1; SMN2KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012085003-A1 2-HYDROXYISOQUINOLINE-1,3(2H,4H)-DIONES AND RELATED COMPOUNDS USEFUL AS HIV REPLICATION INHIBITORS KATHOLIEKE UNIVERSITEIT LEUVEN, K.U. LEUVEN R&D (BE) 2012-06-28 WO disclosed