SCHEMBL10326401

SCHEMBL10326401

CCC(C(=O)O)C1CCN(c2ncc(-c3ccc(C=O)c(F)c3)cc2F)CC1

nearest known ligand 0.39

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MELK Q14680 3/20 0.39
PPARA Q07869 6/20 0.37
PPARG P37231 5/20 0.37
GRIN2B Q13224 4/20 0.37
FFAR4 Q5NUL3 4/20 0.35
ACACB O00763 2/20 0.35
IDO1 P14902 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10324875 0.89 MELK (0.40) MELKGRIN2BFFAR4
SCHEMBL10324422 0.89 DGAT1 (0.43) MELKFFAR4
SCHEMBL10380233 0.80 FFAR4 (0.41) GRIN2BFFAR4
SCHEMBL10380728 0.69 FFAR4 (0.43) GRIN2BFFAR4
SCHEMBL10325542 0.69 GPR119 (0.37)
SCHEMBL17729168 0.69 IDO1 (0.54) IDO1
SCHEMBL10325123 0.66 KDM4E (0.46) MELKGRIN2B
SCHEMBL10326085 0.65 ALOX5AP (0.39) FFAR4
SCHEMBL1976988 0.64 AKR1C3 (0.46)
SCHEMBL21381380 0.63 IDO1 (0.52) IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012096813-A1 IMIDAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2012-07-19 WO disclosed