SCHEMBL10324875

SCHEMBL10324875

CCC(C(=O)O)C1CCN(c2ncc(-c3ccc(C=O)c(F)c3)cn2)CC1

nearest known ligand 0.40

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MELK Q14680 2/20 0.40
AOC3 Q16853 7/20 0.39
TNF P01375 1/20 0.38
FFAR4 Q5NUL3 7/20 0.38
GPR119 Q8TDV5 1/20 0.36
SCD O00767 1/20 0.35
GRIN2B Q13224 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10324422 0.89 DGAT1 (0.43) MELKFFAR4SCD
SCHEMBL10326401 0.89 MELK (0.39) MELKFFAR4GRIN2B
SCHEMBL10380728 0.80 FFAR4 (0.43) AOC3FFAR4GPR119GRIN2B
SCHEMBL10325542 0.78 GPR119 (0.37) AOC3TNFGPR119
SCHEMBL10325755 0.76 AOC3 (0.33) AOC3FFAR4GPR119
SCHEMBL10325123 0.75 KDM4E (0.46) MELKGRIN2B
SCHEMBL17729168 0.69 IDO1 (0.54)
SCHEMBL10380233 0.69 FFAR4 (0.41) FFAR4GRIN2B
SCHEMBL14967451 0.65 GRIN2B (0.41) MELKFFAR4GRIN2B
SCHEMBL1976988 0.64 AKR1C3 (0.46)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012096813-A1 IMIDAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2012-07-19 WO disclosed