SCHEMBL10428536

SCHEMBL10428536

O=C(O)c1c[nH]cc1C(F)(F)F

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 2/20 0.46
ASPH Q12797 1/20 0.44
ALDH1A1 P00352 4/20 0.42
KMT2A Q03164 3/20 0.42
TAS2R14 Q9NYV8 5/20 0.40
FABP4 P15090 1/20 0.39
CLCN2 P51788 1/20 0.37
HPGD P15428 2/20 0.37
KDM4E B2RXH2 1/20 0.37
HSD17B10 Q99714 1/20 0.37
MEN1 O00255 2/20 0.37
CYP1A2 P05177 1/20 0.37
ALOX12 P18054 1/20 0.37
AKR1C3 P42330 1/20 0.36
AKR1C2 P52895 1/20 0.36
DAO P14920 1/20 0.36
CES2 O00748 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL70873 0.77 CFTR (0.50) NOTUMALDH1A1KMT2AKDM4EHSD17B10
SCHEMBL4659258 0.75 GAA (0.40) ALDH1A1KDM4E
SCHEMBL70047 0.74 NOTUM (0.65) NOTUMALDH1A1KMT2AHPGDKDM4E
SCHEMBL7957854 0.74 CES2 (0.31) NOTUMCES2
SCHEMBL1930232 0.74 ALDH1A1 (0.45) NOTUMASPHALDH1A1KMT2AHPGD
SCHEMBL15920412 0.73 ASPH (0.53) NOTUMASPHALDH1A1TAS2R14CLCN2
SCHEMBL3036944 0.73 ASPH (0.59) NOTUMASPHALDH1A1TAS2R14HPGD
SCHEMBL70872 0.72 TAS2R14 (0.41) NOTUMASPHALDH1A1TAS2R14FABP4
SCHEMBL30748715 0.71 ASPH (0.57) NOTUMASPHALDH1A1TAS2R14HPGD
Hydrochloric Acid SCHEMBL22164128 0.71 ASPH (0.57) NOTUMASPHALDH1A1TAS2R14HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101367794-B Preparation method for quinazoline derivants and medical uses thereof SHANGHAI HENGRUI PHARM CO LTD 2013-07-10 CN disclosed
CN-101367794-A Preparation method for quinazoline derivants and medical uses thereof SHANGHAI HENGRUI PHARM CO LTD (CN) 2009-02-18 CN disclosed
EP-0176387-B1 PYRROLE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND THEIR APPLICATION AS PESTICIDES ROUSSEL-UCLAF (FR) 1990-11-22 EP disclosed
EP-0176387-A1 Pyrrole derivatives, process for their preparation and their application as pesticides ROUSSEL-UCLAF (FR) 1986-04-02 EP disclosed