SCHEMBL8317403

SCHEMBL8317403

Cc1ccc(N)c(-c2nc3c(s2)NCCCC3)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 10/20 0.39
BCHE P06276 8/20 0.38
GRIN1 Q05586 7/20 0.38
GRIN2A Q12879 7/20 0.38
TYMS P04818 1/20 0.35
F2RL3 Q96RI0 1/20 0.33
KDM4E B2RXH2 2/20 0.33
NPC1 O15118 2/20 0.33
ALDH1A1 P00352 2/20 0.33
GAA P10253 2/20 0.33
MAPT P10636 2/20 0.33
RAB9A P51151 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
ADORA1 P30542 1/20 0.33
LMNA P02545 1/20 0.32
GLA P06280 1/20 0.32
HPGD P15428 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
PARP1 P09874 1/20 0.31
PARP10 Q53GL7 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10434591 0.84 PDCD1 (0.34) KDM4ENPC1ALDH1A1GAAMAPT
SCHEMBL8316269 0.80 ACHE (0.39) ACHEBCHEGRIN1GRIN2ATYMS
Hydrochloric Acid SCHEMBL8313444 0.80 ALDH1A1 (0.39) ACHEBCHEGRIN1GRIN2AKDM4E
SCHEMBL8315862 0.79 ALOX5 (0.44) KDM4ENPC1ALDH1A1GAAMAPT
SCHEMBL8314378 0.79 RAB9A (0.40) ACHEBCHEGRIN1GRIN2AKDM4E
Hydrochloric Acid SCHEMBL8315136 0.78 ACHE (0.36) ACHEBCHEGRIN1GRIN2AKDM4E
Hydrochloric Acid SCHEMBL8311899 0.78 RAB9A (0.39) ACHEBCHEGRIN1GRIN2AKDM4E
Hydrochloric Acid SCHEMBL8313470 0.77 ACHE (0.40) ACHEBCHEGRIN1GRIN2ATYMS
SCHEMBL8314532 0.76 RAB9A (0.40) ACHEBCHEGRIN1GRIN2AKDM4E
Hydrochloric Acid SCHEMBL8315904 0.75 ACHE (0.39) ACHEBCHEGRIN1GRIN2ATYMS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0351856-B1 Thiazolo[5,4-b]azepine compounds TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1999-09-15 EP disclosed
US-5300639-A 2-oxo-3-carbonylamino-substituted azepine intermediates; lipoperoxide formation inhibitors TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-04-05 US disclosed