SCHEMBL10460244

SCHEMBL10460244

Cc1c(C(=O)[O-])c(=O)cc(-c2ccccc2)n1C.[Na+]

nearest known ligand 0.48

Known targets — ChEMBL curated mechanism

ABCC8ACEADORA1ADORA2AADORA2BADORA3ALDH5A1ALOX5ALOX5APATP4AATP4BBRAFCA1CA12CA2CA4CYSLTR1DHFRDPEP1EDNRAEDNRBESR2F10FDPSFGF1GABBR1GABBR2GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGARTGNRHRGSC1HMGCRIMPDH1IMPDH2KCNJ11LY96NOD2NR3C1NS3NS4ANS5bP2RY1P2RY12P2RY2P2RY4P2RY6PBP2XPDE3APDE3BPDE4APDE4BPDE4CPDE4DPDK1PDK2PDK3PDK4PPARGPPATPTGIRPTGS1PTGS2RAF1RYR1RYR3SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASERPINC1SLC12A1SLC12A3SYKTHRATHRBTLR3TLR4TLR9TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYMSVKORC1XDHblablaIMP-1blaOXA-33blaOXA-58blaT-3blaT-4blaT-5blaT-6dacAdacBdacCfolAfolPfolP1ftsIfusAgaggyrAgyrBmecAmrcAmrcBmrdApbp1apbp1bpbp2pbp2apbp2bpbp3pbp4pbpApbpBpbpCpbpFpolponBrplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpoArpoBrpoCrpoZrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ADORA2B known ✓ P29275 1/20 0.38
HPGD P15428 2/20 0.48
ALDH1A1 P00352 3/20 0.41
KDM4E B2RXH2 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
COMT P21964 1/20 0.40
CYP19A1 P11511 1/20 0.39
MTHFD2 P13995 1/20 0.39
KMT2A Q03164 1/20 0.38
TSHR P16473 1/20 0.38
HSP90AA1 P07900 1/20 0.36
DHODH Q02127 1/20 0.36
PLK1 P53350 1/20 0.36
HTR2A P28223 2/20 0.35
HTR2C P28335 2/20 0.35
SLC6A4 P31645 2/20 0.35
L3MBTL1 Q9Y468 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10463696 0.86 HPGD (0.51) HPGDALDH1A1KDM4ESMN1; SMN2NPSR1
SCHEMBL10460280 0.86 DHODH (0.39) HPGDNPSR1KMT2ADHODH
SCHEMBL10462718 0.86 DHODH (0.39) HPGDALDH1A1KDM4ESMN1; SMN2KMT2A
SCHEMBL10462654 0.85 HPGD (0.48) HPGDALDH1A1KDM4ESMN1; SMN2NPSR1
SCHEMBL10460246 0.85 HPGD (0.50) HPGDALDH1A1KDM4ESMN1; SMN2NPSR1
SCHEMBL10462123 0.82 HPGD (0.43) HPGDALDH1A1KDM4ESMN1; SMN2NPSR1
SCHEMBL10462928 0.80 HPGD (0.46) HPGDALDH1A1KDM4ESMN1; SMN2NPSR1
SCHEMBL10463882 0.79 TSHR (0.58) HPGDALDH1A1KDM4ESMN1; SMN2NPSR1
Hydrochloric Acid SCHEMBL10462633 0.78 TSHR (0.57) HPGDALDH1A1KDM4ESMN1; SMN2NPSR1
SCHEMBL10463752 0.77 COMT (0.42) HPGDALDH1A1KDM4ESMN1; SMN2NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4964896-A GAMETOCIDES MONSANTO COMPANY (US) 1990-10-23 US disclosed
US-4936904-A Aryl-4-oxonicotinates useful for inducing male sterility in cereal grain plants MONSANTO TECHNOLOGY LLC 1990-06-26 US disclosed
US-4714492-A HYBRIDIZATION AGENTS ROHM AND HAAS COMPANY (US) 1987-12-22 US disclosed