Bromide

Bromide

SCHEMBL10550698

CC[c+]1n(N)ccn1CC(=O)c1ccc(Cl)cc1.[Br-]

nearest known ligand 0.45

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHECHKACHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGHRH2OPRM1

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CXCR3 P49682 6/20 0.40
RAB9A P51151 2/20 0.40
GSK3B P49841 2/20 0.39
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA9 Q16790 1/20 0.39
ALDH1A1 P00352 2/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
KDM4E B2RXH2 1/20 0.38
LMNA P02545 1/20 0.38
PKM P14618 1/20 0.37
MAPT P10636 2/20 0.37
MITF O75030 1/20 0.36
S1PR4 O95977 1/20 0.36
TP53 P04637 1/20 0.36
S1PR1 P21453 1/20 0.36
HTT P42858 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL3846592 0.74 CXCR3 (0.44) CXCR3RAB9AGSK3BALDH1A1MEN1
Bromide SCHEMBL10549310 0.74 CXCR3 (0.38) CXCR3RAB9AALDH1A1MEN1KMT2A
SCHEMBL17187853 0.65 GSK3B (0.64) RAB9AGSK3BCA1CA2ALDH1A1
SCHEMBL196299 0.65 GSK3B (0.64) RAB9AGSK3BCA1CA2ALDH1A1
SCHEMBL7214228 0.65 GSK3B (0.64) RAB9AGSK3BCA1CA2ALDH1A1
Bromide SCHEMBL10550683 0.64 PKM (0.44) CXCR3RAB9AGSK3BCA12CA1
SCHEMBL27214768 0.64 RAB9A (0.51) CXCR3RAB9AGSK3BALDH1A1MEN1
SCHEMBL12220178 0.63 GSK3B (0.52) CXCR3RAB9AGSK3BALDH1A1MEN1
Bromide SCHEMBL17180523 0.63 ALDH1A1 (0.61) CXCR3RAB9AGSK3BALDH1A1MEN1
SCHEMBL15340905 0.62 KMT2A (0.64) RAB9AGSK3BALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4831151-A NEMATOCIDES HOFFMANN-LA ROCHE INC. (US) 1989-05-16 US disclosed