SCHEMBL10686151

SCHEMBL10686151

CNS(=O)(=O)c1cc(-c2nc3cnc(OC)nc3[nH]2)c(OC)cc1Cl

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 2/20 0.35
KDR P35968 2/20 0.35
DYRK1A Q13627 2/20 0.35
DYRK1B Q9Y463 2/20 0.35
CDC7 O00311 1/20 0.35
PLK4 O00444 1/20 0.35
CHEK1 O14757 1/20 0.35
AURKA O14965 1/20 0.35
DCLK1 O15075 1/20 0.35
MAPK13 O15264 1/20 0.35
PDPK1 O15530 1/20 0.35
DYRK3 O43781 1/20 0.35
JAK2 O60674 1/20 0.35
ROCK2 O75116 1/20 0.35
RPS6KA5 O75582 1/20 0.35
PRKD3 O94806 1/20 0.35
MAP4K4 O95819 1/20 0.35
PAK4 O96013 1/20 0.35
CHEK2 O96017 1/20 0.35
ABL1 P00519 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10688260 0.89 NR1I2 (0.34) DYRK1ADYRK1BKMT2ASMN1; SMN2PTGES
SCHEMBL10686159 0.84 AURKA (0.35) EGFRKDRDYRK1ADYRK1BCDC7
SCHEMBL10691911 0.81 PKM (0.38) CYP1A2
SCHEMBL10690462 0.78 AMY1A (0.40) SMN1; SMN2POLBAMY1AALDH1A1KDM4E
SCHEMBL10687815 0.77 EGFR (0.37) EGFRKDRDYRK1ADYRK1BCDC7
SCHEMBL10690513 0.75 AMY1A (0.47) PDGFRBPDGFRAMAPK1MAPK8MAPK9
SCHEMBL10686344 0.75 JAK3 (0.35) EGFRKDRDYRK1ADYRK1BCDC7
SCHEMBL10688273 0.72 PDE2A (0.35) AURKATYK2JAK3KMT2ANR1I2
SCHEMBL10690574 0.72 PDE2A (0.51) MAPK1AMY1AALDH1A1KDM4EGAA
SCHEMBL10870043 0.71 MAPT (0.37) DYRK1ADYRK1BPTGESMAPTAMY1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4722929-A Novel 2-phenyl-imidazoles and pharmaceutical compositions containing same DR. KARL THOMAE GMBH (DE) 1988-02-02 US disclosed
EP-0149200-A1 Novel 2-pnenyl-imidazoles, their preparation and drugs containing them Dr. Karl Thomae GmbH (DE) 1985-07-24 EP disclosed