SCHEMBL10691911

SCHEMBL10691911

COc1ncc2nc(-c3cc(S(N)(=O)=O)c(OC)cc3OC)[nH]c2n1

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PKM P14618 2/20 0.38
P2RX3 P56373 2/20 0.36
P2RX2 Q9UBL9 2/20 0.36
PTGES2 Q9H7Z7 2/20 0.36
CA12 O43570 3/20 0.34
CA2 P00918 3/20 0.34
CA9 Q16790 3/20 0.34
CA1 P00915 1/20 0.34
CYP1A2 P05177 2/20 0.33
LDHA P00338 1/20 0.33
PDE5A O76074 1/20 0.32
PDE3B Q13370 1/20 0.32
PDE3A Q14432 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10690462 0.84 AMY1A (0.40) CYP1A2PDE5APDE3BPDE3A
SCHEMBL10688260 0.82 NR1I2 (0.34) CYP1A2
SCHEMBL10691918 0.82 PKM (0.38) PKMP2RX3P2RX2PTGES2CA12
SCHEMBL10686151 0.81 EGFR (0.35) CYP1A2
SCHEMBL10681085 0.78 METAP2 (0.41) PKMP2RX3P2RX2CA12CA2
SCHEMBL10690574 0.75 PDE2A (0.51) CYP1A2PDE5APDE3BPDE3A
SCHEMBL10690513 0.74 AMY1A (0.47) CYP1A2PDE5APDE3BPDE3A
SCHEMBL10689035 0.74 ESR1 (0.42) PDE5APDE3BPDE3A
SCHEMBL10691998 0.72 ADORA2B (0.42) PKMCA12CA2CA9CA1
SCHEMBL10687750 0.71 PKM (0.39) PKMCA12CA2CA9CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4722929-A Novel 2-phenyl-imidazoles and pharmaceutical compositions containing same DR. KARL THOMAE GMBH (DE) 1988-02-02 US disclosed
EP-0149200-A1 Novel 2-pnenyl-imidazoles, their preparation and drugs containing them Dr. Karl Thomae GmbH (DE) 1985-07-24 EP disclosed