SCHEMBL10691729

SCHEMBL10691729

CNS(=O)(=O)c1ccc(-c2nc3c(=O)[nH]ncc3[nH]2)c(OC)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
TAS2R14 Q9NYV8 1/20 0.41
KDM4E B2RXH2 3/20 0.40
ILK Q13418 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
JAK2 O60674 1/20 0.36
JAK1 P23458 1/20 0.36
TYK2 P29597 1/20 0.36
JAK3 P52333 1/20 0.36
PDE5A O76074 1/20 0.36
PDE3B Q13370 1/20 0.36
PDE3A Q14432 1/20 0.36
DHODH Q02127 1/20 0.36
EGFR P00533 1/20 0.35
KDR P35968 1/20 0.35
THRB P10828 1/20 0.35
TNNI3K Q59H18 1/20 0.35
PDE2A O00408 1/20 0.34
HTT P42858 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10686161 0.88 CDK4 (0.42) MEN1KMT2AKDM4EPDE5APDE3B
SCHEMBL10691722 0.87 MEN1 (0.38) MEN1KMT2AKDM4EPDE5APDE3B
SCHEMBL10691563 0.87 CA2 (0.42) MEN1KMT2AKDM4EPDE5APDE3B
SCHEMBL10689653 0.85 MAPT (0.45) MEN1KMT2AKDM4EL3MBTL1PDE5A
SCHEMBL10691045 0.84 TNNI3K (0.41) MEN1KMT2ATAS2R14KDM4EJAK2
SCHEMBL10692684 0.80 ADORA2B (0.46) MEN1KMT2AKDM4EPDE5APDE3B
SCHEMBL10688606 0.80 PDE7A (0.48) PDE5APDE3BPDE3ADHODHPDE2A
SCHEMBL10693845 0.80 GAA (0.43) MEN1KMT2AJAK2JAK1TYK2
SCHEMBL10690895 0.79 TAS2R14 (0.40) MEN1KMT2ATAS2R14KDM4EJAK2
SCHEMBL10686472 0.79 PDE5A (0.37) MEN1KMT2AKDM4EPDE5APDE3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4722929-A Novel 2-phenyl-imidazoles and pharmaceutical compositions containing same DR. KARL THOMAE GMBH (DE) 1988-02-02 US disclosed
EP-0149200-A1 Novel 2-pnenyl-imidazoles, their preparation and drugs containing them Dr. Karl Thomae GmbH (DE) 1985-07-24 EP disclosed