SCHEMBL10692592

SCHEMBL10692592

COc1cccc(C2(Cc3ccccc3)Cc3ccccc3N(C)C2=O)c1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 5/20 0.44
BACE2 Q9Y5Z0 1/20 0.44
AR P10275 2/20 0.41
SCN9A Q15858 1/20 0.41
MEN1 O00255 1/20 0.39
USP2 O75604 1/20 0.39
ALDH1A1 P00352 1/20 0.39
MAPT P10636 1/20 0.39
ALOX15 P16050 1/20 0.39
CASP1 P29466 1/20 0.39
KMT2A Q03164 1/20 0.39
HSD17B10 Q99714 1/20 0.39
CETP P11597 1/20 0.39
SIGMAR1 Q99720 4/20 0.38
POLB P06746 1/20 0.38
PRMT5 O14744 1/20 0.38
WDR77 Q9BQA1 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10693883 0.88 BACE1 (0.44) BACE1BACE2ARSCN9AMEN1
SCHEMBL10695891 0.84 OPRD1 (0.41) AR
SCHEMBL10695992 0.79 SCN9A (0.39) ARSCN9AALDH1A1MAPT
SCHEMBL10692622 0.78 CNR1 (0.39) BACE1AR
SCHEMBL7679980 0.77 BACE1 (0.45) BACE1BACE2ARKMT2ASIGMAR1
SCHEMBL10694802 0.76 BACE1 (0.44) BACE1BACE2SCN9AALDH1A1MAPT
SCHEMBL7677681 0.76 OPRM1 (0.44) BACE1BACE2ARMEN1KMT2A
SCHEMBL10692682 0.74 NPC1 (0.47) BACE1ARUSP2ALDH1A1MAPT
SCHEMBL622589 0.73 PDE4A (0.46) BACE1BACE2ARSCN9AMEN1
SCHEMBL10694576 0.69 POLB (0.33) BACE1ALDH1A1MAPTHSD17B10POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4778793-A CONTROLLING CALCIUM CONCENTRATION-CARDIOVASCULAR DISORDERS HOECHST AKTIENGESELLSCHAFT (DE) 1988-10-18 US disclosed
EP-0212216-A1 Dihydroquinolinone derivatives, processes for their preparation, medicaments containing them, the use of these medicaments, and intermediates for their preparation HOECHST AKTIENGESELLSCHAFT (DE) 1987-03-04 EP disclosed