SCHEMBL10695891

SCHEMBL10695891

CN1C(=O)C(Cc2ccccc2)(c2cccc(O)c2)Cc2ccccc21

nearest known ligand 0.41

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
OPRD1 P41143 13/20 0.41
OPRM1 P35372 10/20 0.39
OPRK1 P41145 9/20 0.39
NR3C1 P04150 1/20 0.37
AR P10275 1/20 0.37
ESR2 Q92731 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10692622 0.87 CNR1 (0.39) NR3C1ARESR2
SCHEMBL10692592 0.84 BACE1 (0.44) AR
SCHEMBL10692682 0.80 NPC1 (0.47) NR3C1AR
SCHEMBL10693883 0.78 BACE1 (0.44) NR3C1AR
SCHEMBL10693819 0.75 OPRD1 (0.40) OPRD1OPRM1OPRK1
SCHEMBL10695992 0.74 SCN9A (0.39) AR
SCHEMBL10694392 0.69 NPC1 (0.47) OPRM1OPRK1
SCHEMBL20714380 0.69 L3MBTL1 (0.41) OPRM1
SCHEMBL10694576 0.68 POLB (0.33)
SCHEMBL980926 0.65 SLC6A2 (0.48)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4778793-A CONTROLLING CALCIUM CONCENTRATION-CARDIOVASCULAR DISORDERS HOECHST AKTIENGESELLSCHAFT (DE) 1988-10-18 US disclosed
EP-0212216-A1 Dihydroquinolinone derivatives, processes for their preparation, medicaments containing them, the use of these medicaments, and intermediates for their preparation HOECHST AKTIENGESELLSCHAFT (DE) 1987-03-04 EP disclosed