SCHEMBL10694802

SCHEMBL10694802

COc1cccc(C2(C(C)C)Cc3ccccc3N(C)C2=O)c1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 7/20 0.44
BACE2 Q9Y5Z0 1/20 0.44
SIGMAR1 Q99720 3/20 0.40
PRMT5 O14744 1/20 0.40
WDR77 Q9BQA1 1/20 0.40
KMT2A Q03164 1/20 0.39
MAPT P10636 1/20 0.39
TSHR P16473 2/20 0.39
SCN9A Q15858 1/20 0.39
ALDH1A1 P00352 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.38
SOAT1 P35610 1/20 0.38
EDNRB P24530 1/20 0.37
EDNRA P25101 1/20 0.37
OPRM1 P35372 1/20 0.37
OPRD1 P41143 1/20 0.37
OPRK1 P41145 1/20 0.37
OPRL1 P41146 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10691593 0.87 L3MBTL1 (0.42) BACE1BACE2KMT2AMAPTTSHR
SCHEMBL10693674 0.84 BACE1 (0.35) BACE1BACE2TSHRALDH1A1
SCHEMBL10693819 0.83 OPRD1 (0.40) SIGMAR1OPRM1OPRD1OPRK1
SCHEMBL10691597 0.77 ADRA1A (0.39) MAPTTSHRSCN9AALDH1A1
SCHEMBL10691351 0.77 GPR55 (0.39) KMT2AMAPTTSHRALDH1A1SMN1; SMN2
SCHEMBL10692592 0.76 BACE1 (0.44) BACE1BACE2SIGMAR1PRMT5WDR77
SCHEMBL10692789 0.73 BACE1 (0.37) BACE1BACE2MAPTTSHRALDH1A1
SCHEMBL10695401 0.72 RAD52 (0.42) BACE1MAPTTSHRALDH1A1OPRM1
SCHEMBL10694665 0.67 RAD52 (0.36) MAPTTSHRALDH1A1OPRM1OPRK1
SCHEMBL10696619 0.65 RAD52 (0.34) MAPTALDH1A1OPRM1OPRK1OPRL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4778793-A CONTROLLING CALCIUM CONCENTRATION-CARDIOVASCULAR DISORDERS HOECHST AKTIENGESELLSCHAFT (DE) 1988-10-18 US disclosed