SCHEMBL10697680

SCHEMBL10697680

Nc1nc(C2=CCN(CCc3ccccc3)CC2)cs1

nearest known ligand 0.67

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.48
DRD4 P21917 2/20 0.48
DRD3 P35462 2/20 0.48
ALDH1A1 P00352 1/20 0.46
MAPT P10636 1/20 0.46
ALOX15 P16050 1/20 0.46
KMT2A Q03164 1/20 0.46
TAAR1 Q96RJ0 1/20 0.46
HSD17B10 Q99714 1/20 0.46
SIGMAR1 Q99720 5/20 0.46
HTR2A P28223 1/20 0.46
HTR2C P28335 1/20 0.46
HTR2B P41595 1/20 0.46
NOS1 P29475 2/20 0.45
LTA4H P09960 1/20 0.43
NOS3 P29474 1/20 0.43
MAOA P21397 1/20 0.42
TMEM97 Q5BJF2 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10697120 0.81 KDM4E (0.42) ALDH1A1MAPTKMT2A
SCHEMBL9451990 0.81 ALDH1A1 (0.46) ALDH1A1MAPTALOX15KMT2ATAAR1
Hydrochloric Acid SCHEMBL10699302 0.80 KDM4E (0.44) ALDH1A1MAPTKMT2A
SCHEMBL10698637 0.79 HTR6 (0.40) SIGMAR1
SCHEMBL30484775 0.77 SIGMAR1 (0.66) DRD2DRD4DRD3SIGMAR1MAOA
Water SCHEMBL10698996 0.77 ALDH1A1 (0.40) DRD2DRD4DRD3ALDH1A1ALOX15
SCHEMBL10332834 0.76 SIGMAR1 (0.53) DRD2DRD4DRD3SIGMAR1
SCHEMBL10698234 0.74 MAPT (0.44) DRD2DRD4DRD3ALDH1A1MAPT
SCHEMBL8583003 0.71 SIGMAR1 (0.52) DRD2DRD4DRD3MAPTSIGMAR1
SCHEMBL6437677 0.71 SIGMAR1 (0.52) DRD2DRD4DRD3SIGMAR1NOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0280873-A1 Piperidines, medicines containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1988-09-07 EP disclosed