SCHEMBL8583003

SCHEMBL8583003

Nc1cc(C2=CCN(CCc3ccccc3)CC2)c[nH]1

nearest known ligand 0.56

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 3/20 0.52
DRD2 P14416 3/20 0.51
DRD4 P21917 3/20 0.51
DRD3 P35462 3/20 0.51
PARP1 P09874 1/20 0.49
HTR1A P08908 2/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
MAPT P10636 1/20 0.47
CYP2C9 P11712 1/20 0.47
TSHR P16473 1/20 0.47
CYP2C19 P33261 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
TMEM97 Q5BJF2 1/20 0.46
S1PR1 P21453 1/20 0.45
S1PR3 Q99500 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30484775 0.83 SIGMAR1 (0.66) SIGMAR1DRD2DRD4DRD3PARP1
SCHEMBL8674007 0.79 SIGMAR1 (0.48) SIGMAR1DRD2DRD4DRD3PARP1
SCHEMBL8585451 0.78 ALOX15 (0.48) DRD2DRD4DRD3HTR1ACYP3A4
SCHEMBL8610590 0.74 SIGMAR1 (0.50) SIGMAR1DRD2DRD4DRD3PARP1
Hydrochloric Acid SCHEMBL11318644 0.73 HTR1A (0.78) SIGMAR1DRD2HTR1ATMEM97
SCHEMBL11329993 0.73 HTR1A (0.78) SIGMAR1DRD2HTR1ATMEM97
SCHEMBL8610861 0.73 L3MBTL1 (0.44) SIGMAR1DRD2DRD4DRD3PARP1
SCHEMBL8584852 0.73 QDPR (0.50) HTR1A
SCHEMBL8194797 0.72 S1PR1 (0.64) SIGMAR1DRD2DRD4DRD3S1PR1
SCHEMBL9501239 0.72 SIGMAR1 (0.55) SIGMAR1DRD2DRD4DRD3PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998020875-A1 5-HT1F AGONISTS ELI LILLY AND COMPANY (US) 1998-05-22 WO disclosed