SCHEMBL10844281

SCHEMBL10844281

[CH2]Cn1nnn(-c2ccccc2)c1=O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.50
ROCK2 O75116 2/20 0.45
ALDH1A1 P00352 8/20 0.40
PKM P14618 2/20 0.40
IDO1 P14902 1/20 0.40
TDO2 P48775 1/20 0.40
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
NPSR1 Q6W5P4 2/20 0.39
GSK3A P49840 1/20 0.38
GSK3B P49841 1/20 0.38
MAPT P10636 3/20 0.38
HTT P42858 2/20 0.38
POLB P06746 2/20 0.37
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C19 P33261 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9779798 0.81 TSHR (0.50) TSHRROCK2ALDH1A1PKMIDO1
SCHEMBL18432812 0.79 ALDH1A1 (0.47) TSHRROCK2ALDH1A1GSK3AGSK3B
SCHEMBL10840968 0.74 IDO1 (0.49) TSHRROCK2ALDH1A1IDO1TDO2
SCHEMBL3521279 0.74 TSHR (0.43) TSHRROCK2ALDH1A1PKMIDO1
SCHEMBL8301872 0.71 ALDH1A1 (0.51) TSHRALDH1A1PKMIDO1TDO2
SCHEMBL8335732 0.71 ADRB2 (0.43) TSHRROCK2ALDH1A1KMT2ANPSR1
SCHEMBL4670086 0.70 ROCK2 (0.61) TSHRROCK2IDO1TDO2CYP1A2
SCHEMBL14600368 0.67 ROCK2 (0.49) TSHRROCK2ALDH1A1PKMIDO1
SCHEMBL4670084 0.66 ROCK2 (0.56) TSHRROCK2ALDH1A1MEN1KMT2A
SCHEMBL4675660 0.66 ROCK2 (0.56) ROCK2ALDH1A1PKMIDO1TDO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4584303-A ANALGESICS THE BOC GROUP, INC. (US) 1986-04-22 US disclosed
EP-0160422-A1 N-Aryl-N-(4-Piperidinyl)amides and pharmaceutical compositions and methods employing such compounds Anaquest, Inc. (US) 1985-11-06 EP disclosed