Triaziquone

Triaziquone

SCHEMBL108508

NC(O)(O)O.O=C1C=C(N2CC2)C(=O)C(N2CC2)=C1N1CC1

nearest known ligand 0.41

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DNMT1 P26358 1/20 0.41
MAPT P10636 2/20 0.39
HTT P42858 2/20 0.39
TP53 P04637 1/20 0.39
STAT3 P40763 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
APAF1 O14727 2/20 0.34
TDP2 O95551 2/20 0.34
NSD2 O96028 2/20 0.34
HKDC1 Q2TB90 2/20 0.34
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
TSHR P16473 1/20 0.33
MAPK1 P28482 1/20 0.33
HIF1A Q16665 1/20 0.33
KMT2A Q03164 2/20 0.33
MEN1 O00255 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Triaziquone SCHEMBL8303 0.88 DNMT1 (0.48) DNMT1MAPTHTTTP53STAT3
Triaziquone SCHEMBL10906735 0.87 HTT (0.43) DNMT1MAPTHTTTP53STAT3
Triaziquone SCHEMBL738610 0.87 DNMT1 (0.42) DNMT1MAPTHTTTP53STAT3
Triaziquone SCHEMBL7783197 0.86 MAPT (0.46) DNMT1MAPTHTTTP53STAT3
Triaziquone SCHEMBL149876 0.86 MAPT (0.46) DNMT1MAPTHTTTP53STAT3
Triaziquone SCHEMBL93807 0.86 DNMT1 (0.37) DNMT1MAPTHTTTP53STAT3
Triaziquone SCHEMBL8482977 0.86 DNMT1 (0.37) DNMT1MAPTHTTTP53STAT3
Triaziquone SCHEMBL6000230 0.86 DNMT1 (0.47) DNMT1MAPTHTTTP53STAT3
Triaziquone SCHEMBL8993238 0.86 DNMT1 (0.47) DNMT1MAPTHTTTP53STAT3
Triaziquone SCHEMBL1538515 0.86 DNMT1 (0.47) DNMT1MAPTHTTTP53STAT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 240 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022268111-A1 ANTIVIRAL PHARMACEUTICAL COMPOSITION, AND PREPARATION METHOD THEREFOR AND APPLICATION THEREOF 前沿生物药业(南京)股份有限公司 2022-12-29 WO claimed
EP-3957627-B1 6-MEMBERED HETEROCYCLIC DERIVATIVE AND PHARMACEUTICAL COMPOSITION COMPRISING SAME SHIONOGI & CO (JP) 2024-06-19 EP disclosed
EP-4219508-B1 SUBSTITUTED POLYCYCLIC PYRIDONE DERIVATIVE AND PRODRUG THEREOF SHIONOGI & CO (JP) 2024-06-05 EP disclosed
EP-4291648-A1 HYBRID AMEBOCYTE LYSATE AND USES THEREOF Charles River Laboratories, Inc. (US) 2023-12-20 EP disclosed
US-11807648-B2 Process for preparing substituted polycyclic pyridone derivative and crystal thereof SHIONOGI & CO., LTD. (JP) 2023-11-07 US disclosed
US-20230287004-A1 SUBSTITUTED POLYCYCLIC PYRIDONE DERIVATIVES AND PRODRUGS THEREOF SHIONOGI & CO., LTD. (JP) 2023-09-14 US disclosed
US-20230258647-A1 HYBRID AMEBOCYTE LYSATE AND USES THEREOF JPMORGAN CHASE BANK, N.A., AS ADMINISTRATIVE AGENT 2023-08-17 US disclosed
EP-4219508-A1 SUBSTITUTED POLYCYCLIC PYRIDONE DERIVATIVE AND PRODRUG THEREOF Shionogi & Co., Ltd (JP) 2023-08-02 EP disclosed
US-20230210822-A1 PHARMACEUTICAL COMPOSITION FOR TREATING FATTY LIVER DISEASE SHIONOGI & CO., LTD. (JP) 2023-07-06 US disclosed
EP-4194459-A1 PROCESS FOR PREPARING SUBSTITUTED POLYCYCLIC PYRIDONE DERIVATIVE AND CRYSTAL THEREOF Shionogi & Co., Ltd (JP) 2023-06-14 EP disclosed
US-5523077-A CONTAINING BUTHIONINE SULFOXIMINE OR CYSTAMINE AND HYDROQUINONE OR ETHER THEREOF YALE UNIVERSITY (US) 1996-06-04 US disclosed
EP-0688204-A1 COMPOSITION AND METHOD FOR WHITENING SKIN YALE UNIVERSITY (US) 1995-12-27 EP disclosed
WO-1994020068-A1 COMPOSITION AND METHOD FOR WHITENING SKIN YALE UNIVERSITY (US) 1994-09-15 WO disclosed
US-5310657-A Monitoring absorption spectra, analysis of water systems, body fluids WHITTAKER BIOPRODUCTS, INC. (US) 1994-05-10 US disclosed
EP-0426395-A1 Kinetic assay for endotoxin using limulus amebocyte lysate and chromogenic substrate BIOWHITTAKER, INC. (US) 1991-05-08 EP disclosed
EP-0096074-A4 EXPANDABLE LATTICE OF POLYVINYL ALCOHOL AND POLYETHYLENE GLYCOL. KEY PHARMA (US) 1984-05-29 EP disclosed
US-4428925-A LATTICE COATING OF POLYVINYL ALCOHOL AND POLYOXYETHYLENE GLYCOL KEY PHARMACEUTICALS, INC. (US) 1984-01-31 US disclosed
US-4428926-A LATTICE COATING OF POLYVINYL ALCOHOL AND POLYOXYETHYLENE GLYCOL KEY PHARMACEUTICALS, INC. (US) 1984-01-31 US disclosed
EP-0096074-A1 EXPANDABLE LATTICE OF POLYVINYL ALCOHOL AND POLYETHYLENE GLYCOL Key Pharmaceuticals, Inc. (US) 1983-12-21 EP disclosed
WO-1983002056-A1 EXPANDABLE LATTICE OF POLYVINYL ALCOHOL AND POLYETHYLENE GLYCOL KEY PHARMA (US) 1983-06-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11807648-B2 Process for preparing substituted polycyclic pyridone derivative and crystal thereof REN, C5, PDXK DNMT1 1010/4885MAPT 3290/4885HTT 2614/4885
US-20230287004-A1 SUBSTITUTED POLYCYCLIC PYRIDONE DERIVATIVES AND PRODRUGS THEREOF C3AR1, NR4A1, HAVCR2 DNMT1 1796/4885MAPT 4872/4885HTT 4544/4885
US-20230210822-A1 PHARMACEUTICAL COMPOSITION FOR TREATING FATTY LIVER DISEASE LIPC, PNLIP, ACACB DNMT1 4865/4885MAPT 4017/4885HTT 1614/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.