SCHEMBL10969348

SCHEMBL10969348

O=C1CC=CC2=C1Nc1ccccc1CN2

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR5A P47898 4/20 0.41
AHR P35869 1/20 0.39
PDK2 Q15119 1/20 0.39
BRD4 O60885 2/20 0.38
CREBBP Q92793 2/20 0.38
NPC1 O15118 2/20 0.38
MAPK13 O15264 1/20 0.38
MAPK12 P53778 1/20 0.38
MAPK11 Q15759 1/20 0.38
MAPK14 Q16539 1/20 0.38
MAPT P10636 2/20 0.36
CA12 O43570 1/20 0.35
CA9 Q16790 1/20 0.35
ALOX15 P16050 1/20 0.35
HSD17B10 Q99714 1/20 0.35
GAA P10253 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
KDM4E B2RXH2 1/20 0.32
MEN1 O00255 1/20 0.32
HSP90AA1 P07900 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28517190 0.82 PDGFRA (0.35) AHRPDK2BRD4CREBBPNPC1
SCHEMBL28552531 0.73 AHR (0.50) HTR5AAHRPDK2BRD4CREBBP
SCHEMBL6775003 0.72 CA12 (0.49) CA12CA9KDM4E
SCHEMBL8872856 0.71 CA12 (0.55) HTR5AAHRPDK2BRD4CREBBP
SCHEMBL7982185 0.70 MEN1 (0.48) AHRPDK2BRD4CREBBPNPC1
SCHEMBL45104 0.69 HTR5A (0.53) HTR5AAHRPDK2BRD4CREBBP
SCHEMBL6136738 0.66 AHR (0.48) HTR5AAHRPDK2BRD4CREBBP
SCHEMBL9211112 0.65 ALOX5 (0.44) BRD4CREBBPMAPTGAANPSR1
SCHEMBL310398 0.65 HTR5A (0.57) HTR5AAHRPDK2BRD4CREBBP
SCHEMBL9094422 0.64 AHR (0.40) AHRPDK2BRD4CREBBPNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4556653-A ANTISECRETORY, ANTIULCER AND ANTISPASMODIC AGENTS DOMPE' FARMACEUTICA S.P.A. (IT) 1985-12-03 US disclosed