SCHEMBL11021091

SCHEMBL11021091

CCOc1cc(S(N)(=O)=O)ccc1-c1nc2ccc(C#N)cc2[nH]1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATR Q13535 1/20 0.48
CA12 O43570 2/20 0.43
CA1 P00915 2/20 0.43
CA2 P00918 2/20 0.43
CA9 Q16790 2/20 0.43
CA3 P07451 1/20 0.43
CA4 P22748 1/20 0.43
CA6 P23280 1/20 0.43
CA5A P35218 1/20 0.43
CA7 P43166 1/20 0.43
CA14 Q9ULX7 1/20 0.43
CA5B Q9Y2D0 1/20 0.43
METAP2 P50579 1/20 0.43
METAP1 P53582 1/20 0.43
PKN1 Q16512 1/20 0.43
PKN2 Q16513 1/20 0.43
CHEK2 O96017 5/20 0.42
SCD O00767 1/20 0.41
MAPT P10636 3/20 0.41
TTK P33981 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11021081 0.92 CA12 (0.43) ATRCA12CA1CA2CA9
SCHEMBL11022217 0.91 ATR (0.53) ATRMETAP2METAP1PKN1PKN2
SCHEMBL11020318 0.89 CA12 (0.54) ATRCA12CA1CA2CA9
SCHEMBL11021741 0.88 ATR (0.44) ATRMETAP2METAP1PKN1PKN2
SCHEMBL11021240 0.88 MAPT (0.46) ATRMETAP2METAP1PKN1PKN2
SCHEMBL11022213 0.83 ATR (0.44) ATRSCDMAPTTRPV4
SCHEMBL11018186 0.82 CYP3A4 (0.48) ATRPKN1PKN2SCD
SCHEMBL11018070 0.81 METAP2 (0.44) ATRMETAP2METAP1PKN1PKN2
SCHEMBL11020313 0.81 CA2 (0.54) ATRCA12CA1CA2CA9
SCHEMBL11021674 0.81 METAP2 (0.46) ATRMETAP2METAP1PKN1PKN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0148431-A1 Benzimidazoles, their preparation, and medicaments containing these compounds Dr. Karl Thomae GmbH (DE) 1985-07-17 EP disclosed