SCHEMBL11050004

SCHEMBL11050004

CC(C)(C)NC(=O)NC(=N)Nc1ccc(C(F)(F)F)cc1Cl

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.47
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
CA9 Q16790 1/20 0.47
ALDH1A1 P00352 3/20 0.47
MAPT P10636 1/20 0.47
IDH1 O75874 1/20 0.45
HTT P42858 1/20 0.44
ACHE P22303 1/20 0.42
SMO Q99835 1/20 0.41
KDR P35968 2/20 0.41
NTRK1 P04629 2/20 0.41
RET P07949 1/20 0.41
PDGFRB P09619 1/20 0.41
PDGFRA P16234 1/20 0.41
CDK8 P49336 1/20 0.41
NTRK3 Q16288 1/20 0.41
MAPK14 Q16539 1/20 0.41
NTRK2 Q16620 1/20 0.41
MEN1 O00255 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11049781 0.88 KIF11 (0.46) CA12CA1CA2CA9HTT
SCHEMBL11255956 0.87 MEN1 (0.42) MAPTIDH1HTTNTRK1NTRK2
SCHEMBL11052904 0.86 HTT (0.47) HTTMEN1KMT2APOLBMAPK1
SCHEMBL11053855 0.85 MAPT (0.40) CA12CA1CA2CA9ALDH1A1
SCHEMBL11250280 0.85 LMNA (0.41) MAPTHTTMEN1KMT2ALMNA
SCHEMBL11052114 0.84 PDK1 (0.50) ALDH1A1MAPTHTTMEN1KMT2A
SCHEMBL11261823 0.84 TAS2R14 (0.44) ALDH1A1MAPTIDH1HTTKDR
SCHEMBL11059026 0.83 RAB9A (0.47) ALDH1A1MAPTHTTMEN1KMT2A
SCHEMBL11048661 0.82 MAPK1 (0.52) ALDH1A1MAPTHTTMEN1KMT2A
SCHEMBL11048648 0.82 HTT (0.43) ALDH1A1MAPTHTTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4488993-A Amidinoureas WILLIAM H. RORER, INC. 1984-12-18 US disclosed
US-4220658-A Treatment of hypertension with amidinoureas WILLIAM H. RORER, INC. (US) 1980-09-02 US disclosed
US-4088785-A HYPOTENSIVE AGENTS WILLIAM H. RORER, INC. (US) 1978-05-09 US disclosed