SCHEMBL11059402

SCHEMBL11059402

CCOc1cccc(C)c1-n1cnc(NC)nc1=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.39
MAPT P10636 4/20 0.39
MEN1 O00255 3/20 0.39
L3MBTL1 Q9Y468 3/20 0.39
KDM4E B2RXH2 2/20 0.39
LMNA P02545 2/20 0.39
POLB P06746 1/20 0.39
GAA P10253 1/20 0.39
RECQL P46063 1/20 0.39
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
HCAR1 Q9BXC0 1/20 0.35
TP53 P04637 5/20 0.35
PKM P14618 1/20 0.34
GRK6 P43250 2/20 0.34
PABPC1 P11940 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
ELANE P08246 1/20 0.34
GRM5 P41594 1/20 0.33
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11058341 0.88 APLNR (0.38) KMT2AMAPTMEN1L3MBTL1KDM4E
SCHEMBL11054404 0.86 HCAR1 (0.46) KMT2AMEN1POLBHCAR1ELANE
SCHEMBL11059212 0.85 HCAR1 (0.38) KMT2AMEN1POLBHCAR1TP53
Hydrochloric Acid SCHEMBL11052665 0.84 HCAR1 (0.44) KMT2AMEN1POLBHCAR1ELANE
SCHEMBL11054891 0.82 PKM (0.41) KMT2AMAPTMEN1L3MBTL1KDM4E
SCHEMBL11057854 0.80 HCAR1 (0.41) KMT2AMEN1LMNAPOLBHCAR1
SCHEMBL11054879 0.80 HCAR1 (0.38) POLBHCAR1ELANE
SCHEMBL11050172 0.80 HCAR1 (0.38) HCAR1
SCHEMBL11054604 0.80 CHRNA7 (0.47) HCAR1
SCHEMBL11057840 0.79 FGFR1 (0.36) KMT2AMAPTMEN1L3MBTL1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4452980-A DIARRHEA WILLIAM H. RORER, INC. (US) 1984-06-05 US disclosed
US-4246409-A ANTIDIARRHEAL AGENTS WILLIAM H. RORER, INC. (US) 1981-01-20 US disclosed
US-4225315-A Triazinones from amidinoureas WILLIAM H. RORER, INC. (US) 1980-09-30 US disclosed