SCHEMBL11063299

SCHEMBL11063299

CCOC(=O)Cc1c(C(=O)OCC)c2c(n1C)-c1c(cc(Cl)ccc1=O)CC2

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.38
ALOX15 P16050 2/20 0.38
TSHR P16473 2/20 0.38
HSD17B10 Q99714 2/20 0.38
KDM4E B2RXH2 1/20 0.38
HPGD P15428 1/20 0.38
CASP1 P29466 1/20 0.38
GABRA1 P14867 1/20 0.36
GABRG2 P18507 1/20 0.36
GABRB3 P28472 1/20 0.36
GABRA5 P31644 1/20 0.36
GABRA3 P34903 1/20 0.36
GABRA2 P47869 1/20 0.36
GABRB2 P47870 1/20 0.36
GABRA4 P48169 1/20 0.36
GABRA6 Q16445 1/20 0.36
KDM1A O60341 1/20 0.36
LMNA P02545 4/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
CYP1A2 P05177 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11060030 0.92 LMNA (0.36) ALDH1A1ALOX15TSHRHSD17B10KDM4E
SCHEMBL11066911 0.87 KDM1A (0.41) ALDH1A1ALOX15TSHRHSD17B10KDM4E
SCHEMBL11072105 0.81 SRD5A1 (0.35) L3MBTL1
SCHEMBL11062697 0.80 LMNA (0.40) ALDH1A1ALOX15TSHRHSD17B10KDM4E
SCHEMBL11065609 0.80 HRH1 (0.39) ALDH1A1ALOX15TSHRHSD17B10KDM4E
SCHEMBL11068485 0.77 L3MBTL1 (0.42) ALDH1A1KDM4EKDM1ALMNAL3MBTL1
SCHEMBL11066786 0.77 ALDH1A1 (0.45) ALDH1A1KDM4EHPGDKDM1ALMNA
SCHEMBL11071003 0.76 MAPK14 (0.42) ALDH1A1TSHRGABRA1GABRG2GABRB3
SCHEMBL11186665 0.75 KDM1A (0.36) ALDH1A1TSHRHSD17B10KDM4EHPGD
SCHEMBL11063136 0.75 PTGDR2 (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4440779-A Tricyclic derivatives of substituted pyrrole acids as analgesic and anti-inflammatory agents MERCK & CO., INC. (US) 1984-04-03 US disclosed
EP-0068460-A1 Tricyclic derivatives of substituted pyrrole acids as analgesic and anti-inflammatory agents MERCK & CO. INC. (US) 1983-01-05 EP disclosed