SCHEMBL11270864

SCHEMBL11270864

COc1ccc(CN2C3CCC2CC(C(=O)Nc2cc(Cl)c(NC=O)cc2OC)C3)cc1

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 1/20 0.46
TSHR P16473 1/20 0.43
L3MBTL1 Q9Y468 3/20 0.43
LTA4H P09960 1/20 0.43
ALPL P05186 1/20 0.42
ALPI P09923 1/20 0.42
ALPG P10696 1/20 0.42
ALDH1A1 P00352 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C19 P33261 1/20 0.41
SIGMAR1 Q99720 1/20 0.41
DRD4 P21917 2/20 0.40
DRD3 P35462 1/20 0.40
CHEK1 O14757 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11093528 0.94 CXCR6 (0.47) TSHRSIGMAR1DRD4DRD3
SCHEMBL11094396 0.93 SIGMAR1 (0.46) TSHRSIGMAR1DRD4DRD3
SCHEMBL11097362 0.92 TSHR (0.43) TSHRSIGMAR1DRD4DRD3
SCHEMBL11097324 0.92 DRD4 (0.48) TSHRDRD4DRD3
SCHEMBL11270191 0.89 CXCR4 (0.47) CXCR4TSHRL3MBTL1LTA4HALPL
SCHEMBL11097949 0.86 DRD2 (0.51) CXCR4TSHRL3MBTL1LTA4HALPL
SCHEMBL11095214 0.85 UBE2M (0.44) TSHRALDH1A1SIGMAR1DRD4DRD3
SCHEMBL11100155 0.84 OPRM1 (0.45) TSHRL3MBTL1ALPLALPIALPG
SCHEMBL11096161 0.84 DRD4 (0.51) TSHRDRD4DRD3
SCHEMBL11089660 0.84 HCRTR1 (0.53) CXCR4TSHRALDH1A1SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0031219-A1 Aniline derivatives BEECHAM GROUP PLC (GB) 1981-07-01 EP claimed
US-4350691-A ANTIEMETICS BEECHAM GROUP LIMITED (GB) 1982-09-21 US disclosed
EP-0031219-A1 Aniline derivatives BEECHAM GROUP PLC (GB) 1981-07-01 EP disclosed