SCHEMBL11101044

SCHEMBL11101044

CCS(=O)(=O)c1ccc(-n2ccccc2=O)cc1

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PSIP1 O75475 2/20 0.52
GAA P10253 1/20 0.43
APLNR P35414 4/20 0.40
F10 P00742 7/20 0.38
F2 P00734 1/20 0.38
F11 P03951 1/20 0.38
PTGS2 P35354 2/20 0.37
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA9 Q16790 1/20 0.37
CA14 Q9ULX7 1/20 0.37
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
CYP1A2 P05177 1/20 0.36
HPGD P15428 1/20 0.36
BLM P54132 1/20 0.36
HSD17B10 Q99714 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1381320 0.82 PTGS2 (0.53) F10PTGS2
SCHEMBL10059528 0.79 CA12 (0.54) PTGS2CA12CA1CA2CA9
SCHEMBL14490265 0.77 MGLL (0.48) GAAF10KDM4EALDH1A1CYP1A2
SCHEMBL14502379 0.75 F10 (0.49) GAAF10ALDH1A1
SCHEMBL92819 0.74 KDM4E (0.57) F10F2CA1CA2KDM4E
SCHEMBL4694832 0.72 F10 (0.49) GAAF10F2ALDH1A1
SCHEMBL143175 0.72 ALDH1A1 (0.54) GAAF10KDM4EALDH1A1CYP1A2
SCHEMBL10455034 0.72 PSIP1 (0.74) PSIP1GAACA2ALDH1A1
SCHEMBL2645575 0.71 DDB1 (0.41) F10CA12CA1CA2CA9
SCHEMBL28203632 0.71 KEAP1 (0.53) F10PTGS2CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4517192-A 6-Alkyl-5-[4-(alkylsulfinyl or alkylsulfonyl)phenyl]-2(1H)-pyridinones and their use as cardiatonics STERLING DRUG INC. (US) 1985-05-14 US disclosed