SCHEMBL1114262

SCHEMBL1114262

CCC(C)Nc1c(S(N)(=O)=O)ccc(Sc2ccccc2)c1[N+](=O)[O-]

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 10/20 0.40
CA4 P22748 10/20 0.40
CA12 O43570 8/20 0.38
CA1 P00915 8/20 0.38
CA3 P07451 8/20 0.38
CA6 P23280 8/20 0.38
CA7 P43166 8/20 0.38
CA9 Q16790 8/20 0.38
CA13 Q8N1Q1 8/20 0.38
CA14 Q9ULX7 8/20 0.38
CA5B Q9Y2D0 8/20 0.38
CA5A P35218 7/20 0.38
ALDH1A1 P00352 2/20 0.38
CYP1A2 P05177 2/20 0.38
CYP2C19 P33261 2/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
HTT P42858 1/20 0.38
MAPT P10636 3/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4215302 0.89 HTT (0.42) CA2CA4CA12CA1CA3
SCHEMBL1114369 0.81 HTT (0.44) CA2CA4ALDH1A1CYP1A2CYP2C19
SCHEMBL4219323 0.73 CA12 (0.37) CA2CA4CA12CA6CA7
SCHEMBL6468837 0.73 CA2 (0.38) CA2CA4CA12CA1CA3
SCHEMBL1114110 0.71 CA2 (0.36) CA2CA4CA12CA1CA3
SCHEMBL11677839 0.68 ALDH1A1 (0.58) ALDH1A1CYP1A2CYP2C19CYP3A4CYP2C9
SCHEMBL8433529 0.65 L3MBTL1 (0.39) ALDH1A1CYP1A2CYP2C19CYP3A4CYP2C9
SCHEMBL6025517 0.63 KMT2A (0.44) CA2CA1CA9ALDH1A1MAPT
SCHEMBL4707544 0.63 PDE7A (0.48) ALDH1A1CYP3A4HTTMAPTGAA
SCHEMBL6530527 0.62 KMT2A (0.41) CA2CA9ALDH1A1CYP2C19CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2279174-A2 ARYLSULFONAMIDE COMPOUNDS, COMPOSITIONS AND METHODS OF USE Genentech, Inc. (US) 2011-02-02 EP disclosed
WO-2009143246-A2 ARYLSULFONAMIDE COMPOUNDS, COMPOSITIONS AND METHODS OF USE GENENTECH, INC. (US) 2009-11-26 WO disclosed
WO-2005049593-A2 N-ACYLSULFONAMIDE APOPTOSIS PROMOTERS ABBOTT LABORATORIES (US) 2005-06-02 WO disclosed