SCHEMBL11204668

SCHEMBL11204668

CNc1[nH]c2cc(N3CCC(O)CC3)c(F)cc2c(=O)c1C(=O)O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 2/20 0.40
GSK3A P49840 2/20 0.40
GSK3B P49841 2/20 0.40
PIM3 Q86V86 2/20 0.40
PRKD3 O94806 1/20 0.40
IRAK1 P51617 1/20 0.40
RPS6KA3 P51812 1/20 0.40
DYRK1A Q13627 1/20 0.40
CSNK1G3 Q9Y6M4 1/20 0.40
ALDH1A1 P00352 6/20 0.38
LMNA P02545 6/20 0.38
KDM4E B2RXH2 5/20 0.38
HPGD P15428 4/20 0.38
HSD17B10 Q99714 4/20 0.38
CYP1A2 P05177 1/20 0.38
TOP2A P11388 1/20 0.38
CYP2C9 P11712 1/20 0.38
TOP2B Q02880 1/20 0.38
MAPT P10636 1/20 0.37
BRD4 O60885 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11205213 0.94 PIM1 (0.42) PIM1GSK3AGSK3BPIM3PRKD3
SCHEMBL11204174 0.87 ALDH1A1 (0.47) ALDH1A1LMNAKDM4EHPGDHSD17B10
SCHEMBL11203701 0.86 HPGD (0.43) ALDH1A1LMNAKDM4EHPGDHSD17B10
SCHEMBL11199207 0.84 ALDH1A1 (0.48) ALDH1A1LMNAKDM4EHPGDHSD17B10
SCHEMBL11209760 0.83 DRD3 (0.41) ALDH1A1LMNAKDM4EHPGDHSD17B10
SCHEMBL11203471 0.75 GPR84 (0.38) ALDH1A1KDM4E
SCHEMBL11208613 0.74 GAA (0.47) ALDH1A1KDM4EHPGDHSD17B10MAPT
SCHEMBL7557799 0.72 ALDH1A1 (0.51) PIM1GSK3AGSK3BPIM3PRKD3
SCHEMBL3474228 0.70 ALDH1A1 (0.53) ALDH1A1LMNAKDM4EHPGDHSD17B10
SCHEMBL9523388 0.70 LMNA (0.64) PIM1GSK3AGSK3BPIM3PRKD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0090424-A1 New quinolone compounds and preparation thereof STERLING DRUG INC. (US) 1983-10-05 EP disclosed