SCHEMBL11205751

SCHEMBL11205751

CN(C)C(=O)C(C#N)(Sc1ccccc1)Sc1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 4/20 0.41
OPRM1 P35372 4/20 0.41
DRD3 P35462 4/20 0.41
DRD2 P14416 3/20 0.38
ALDH1A1 P00352 4/20 0.37
SMN1; SMN2 Q16637 3/20 0.37
RAB9A P51151 3/20 0.37
KMT2A Q03164 3/20 0.37
MEN1 O00255 2/20 0.37
NPSR1 Q6W5P4 2/20 0.35
LMNA P02545 2/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
CYP3A4 P08684 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
HPGD P15428 2/20 0.33
CYP2D6 P10635 1/20 0.33
ABCC9 O60706 1/20 0.32
ABCC8 Q09428 1/20 0.32
KCNJ11 Q14654 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11205161 0.86 KMT2A (0.38) ALDH1A1SMN1; SMN2RAB9AKMT2AMEN1
SCHEMBL11268140 0.80 FFAR1 (0.36) ALDH1A1SMN1; SMN2RAB9AKMT2ANPSR1
SCHEMBL11265046 0.79 MAPT (0.38) ALDH1A1KMT2ALMNAL3MBTL1CYP3A4
SCHEMBL11271178 0.72 TGM2 (0.43) ALDH1A1SMN1; SMN2RAB9AKMT2AMEN1
SCHEMBL11202360 0.72 LMNA (0.36) ALDH1A1SMN1; SMN2RAB9AKMT2AMEN1
SCHEMBL9268675 0.70 OPRM1 (0.47) DRD4OPRM1DRD3DRD2ALDH1A1
SCHEMBL11260235 0.68 ALDH1A1 (0.47) ALDH1A1SMN1; SMN2RAB9AKMT2AMEN1
SCHEMBL9268779 0.68 OPRM1 (0.45) DRD4OPRM1DRD3DRD2ALDH1A1
SCHEMBL2951109 0.68 MAOA (0.40) DRD4OPRM1DRD3DRD2ALDH1A1
SCHEMBL10346433 0.67 OPRM1 (0.44) DRD4OPRM1DRD3DRD2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0029719-B1 VULCANIZABLE RUBBER COMPOSITIONS INHIBITED FROM PREMATURE VULCANIZATION BY METHYLENE THIOETHERS, AND NOVEL METHYLENE THIOETHERS MONSANTO COMPANY (US) 1983-02-16 EP disclosed
US-4342705-A CONTAINING CARBONYL OR CYANO FUNCTIONAL GROUPS, USEFUL AS VULCANIZATION INHIBITORS MONSANTO COMPANY (US) 1982-08-03 US disclosed
EP-0029719-A1 Vulcanizable rubber compositions inhibited from premature vulcanization by methylene thioethers, and novel methylene thioethers MONSANTO COMPANY (US) 1981-06-03 EP disclosed
US-4271050-A Vulcanizable rubber compositions inhibited from premature vulcanization by methylene thioethers MONSANTO COMPANY (US) 1981-06-02 US disclosed