SCHEMBL11218549

SCHEMBL11218549

Cc1nc(-c2ccccc2)c[n+]([O-])c1N

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
ADORA2A P29274 3/20 0.41
ADORA1 P30542 3/20 0.41
ALDH1A1 P00352 4/20 0.41
NPC1 O15118 2/20 0.41
HPGD P15428 1/20 0.41
NFKB1 P19838 1/20 0.41
HTT P42858 1/20 0.41
NFKB2 Q00653 1/20 0.41
RELA Q04206 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
ASIC3 Q9UHC3 1/20 0.40
KDM4E B2RXH2 1/20 0.39
MAPT P10636 1/20 0.39
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA7 P43166 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7107176 0.78 ADORA1 (0.43) RAB9AMEN1KMT2AADORA2AADORA1
SCHEMBL9791429 0.75 KDM4E (0.47) RAB9AMEN1KMT2AALDH1A1HPGD
SCHEMBL11227298 0.74 ADORA2A (0.41) RAB9AMEN1KMT2AADORA2AADORA1
SCHEMBL2659278 0.70 KMT2A (0.42) RAB9AMEN1KMT2AALDH1A1NPC1
SCHEMBL4906692 0.70 SMN1; SMN2 (0.42) RAB9AMEN1KMT2AALDH1A1NPC1
SCHEMBL6618672 0.69 ALDH1A1 (0.55) RAB9AMEN1KMT2AADORA2AADORA1
SCHEMBL1752891 0.67 RAB9A (0.42) RAB9AMEN1KMT2AALDH1A1NPC1
SCHEMBL864957 0.67 ASIC3 (0.47) RAB9AMEN1KMT2AADORA2AADORA1
SCHEMBL8012385 0.67 ACHE (0.55) RAB9AMEN1KMT2AADORA2AADORA1
SCHEMBL2681285 0.67 SMN1; SMN2 (0.51) RAB9AADORA2AADORA1ALDH1A1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4343802-A ADRENERGIC BLOCKING, ANTIARRYHYTHMIA, AND CARDIOTONIC AGENTS MERCK, SHARP & DOHME (I.A.) CORP. (US) 1982-08-10 US disclosed
US-4193995-A B-ADRENERGIC BLOCKING AGENTS MERCK SHARP & DOHME (I.A.) CORP. (US) 1980-03-18 US disclosed
US-4042586-A ADRENERGIC BLOCKING AGENTS MERCK SHARP & DOHME (I.A.) CORPORATION (US) 1977-08-16 US disclosed
US-3946009-A ADRENERGIC BLOCKING AGENTS MERCK SHARP & DOHME (I.A.) CORPORATION (US) 1976-03-23 US disclosed