SCHEMBL11240925

SCHEMBL11240925

O=C(O)Cc1ccc2c(c1)sc1cccc(Cl)c12

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SLC22A12 Q96S37 12/20 0.46
MAPK1 P28482 1/20 0.46
MCL1 Q07820 1/20 0.46
CA2 P00918 1/20 0.45
AKR1B1 P15121 1/20 0.42
OGG1 O15527 1/20 0.42
GAA P10253 1/20 0.40
KDM4E B2RXH2 1/20 0.40
THRA P10827 1/20 0.40
THRB P10828 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11239805 0.84 CA2 (0.46) SLC22A12MCL1CA2AKR1B1GAA
SCHEMBL11228298 0.82 CA2 (0.50) SLC22A12MCL1CA2AKR1B1GAA
SCHEMBL11228323 0.82 L3MBTL1 (0.49) SLC22A12MAPK1MCL1OGG1GAA
SCHEMBL11228329 0.81 CA2 (0.43) SLC22A12MCL1CA2KDM4E
SCHEMBL11242747 0.81 CA2 (0.45) SLC22A12CA2AKR1B1GAAKDM4E
SCHEMBL11232390 0.79 AKR1B1 (0.53) AKR1B1GAAKDM4E
SCHEMBL11242088 0.78 BCKDK (0.51) SLC22A12MAPK1MCL1CA2AKR1B1
Methane SCHEMBL11248449 0.78 AKR1B1 (0.51) AKR1B1GAAKDM4E
SCHEMBL11246405 0.76 BCL2L1 (0.50) SLC22A12MCL1AKR1B1GAAKDM4E
SCHEMBL26312266 0.75 AKR1B1 (0.60) AKR1B1GAAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4334078-A ANTIINFLAMMATORY AGENTS, ANALGESICS, ANTIRHEUMATICS HOFFMANN-LA ROCHE INC. (US) 1982-06-08 US disclosed
US-4219657-A USED AS ANTIINFLAMATORY AGENTS, ANALGESICS, ANTIRHEUMATIC AGENTS HOFFMANN-LA ROCHE INC. (US) 1980-08-26 US disclosed