SCHEMBL11242747

SCHEMBL11242747

O=C(O)Cc1ccc2c(c1)sc1c(Cl)cccc12

nearest known ligand 0.45

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CA2 P00918 1/20 0.45
SLC22A12 Q96S37 11/20 0.44
AKR1B1 P15121 2/20 0.43
KDM4E B2RXH2 2/20 0.42
ALDH1A1 P00352 1/20 0.42
HPGD P15428 1/20 0.42
HSD17B10 Q99714 1/20 0.42
THRA P10827 1/20 0.41
THRB P10828 1/20 0.41
GAA P10253 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11243751 0.84 CA2 (0.46) CA2SLC22A12AKR1B1KDM4EALDH1A1
SCHEMBL11236198 0.82 L3MBTL1 (0.46) KDM4EALDH1A1GAA
SCHEMBL11240925 0.81 SLC22A12 (0.46) CA2SLC22A12AKR1B1KDM4ETHRA
SCHEMBL11228298 0.80 CA2 (0.50) CA2SLC22A12AKR1B1KDM4EALDH1A1
SCHEMBL11232390 0.79 AKR1B1 (0.53) AKR1B1KDM4EALDH1A1HPGDHSD17B10
Methane SCHEMBL11248449 0.78 AKR1B1 (0.51) AKR1B1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL11242088 0.78 BCKDK (0.51) CA2SLC22A12AKR1B1KDM4EALDH1A1
SCHEMBL11246405 0.76 BCL2L1 (0.50) SLC22A12AKR1B1KDM4EALDH1A1HPGD
SCHEMBL11244597 0.75 CA2 (0.45) CA2SLC22A12KDM4EALDH1A1HPGD
SCHEMBL11240017 0.74 KEAP1 (0.51) CA2SLC22A12KDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4334078-A ANTIINFLAMMATORY AGENTS, ANALGESICS, ANTIRHEUMATICS HOFFMANN-LA ROCHE INC. (US) 1982-06-08 US disclosed
US-4219657-A USED AS ANTIINFLAMATORY AGENTS, ANALGESICS, ANTIRHEUMATIC AGENTS HOFFMANN-LA ROCHE INC. (US) 1980-08-26 US disclosed