SCHEMBL11241215

SCHEMBL11241215

CC(C)(C)c1nc(Cl)c(Br)cc1-c1ccncc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 2/20 0.37
S1PR1 P21453 1/20 0.36
S1PR3 Q99500 1/20 0.36
TRPV1 Q8NER1 2/20 0.35
GCGR P47871 5/20 0.35
MAPK14 Q16539 3/20 0.34
NPC1 O15118 3/20 0.34
RAB9A P51151 3/20 0.34
HTT P42858 2/20 0.34
MAPT P10636 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
LMNA P02545 1/20 0.34
TP53 P04637 1/20 0.34
HPGD P15428 1/20 0.34
TSHR P16473 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
BRAF P15056 1/20 0.34
PDE3B Q13370 2/20 0.33
PDE3A Q14432 2/20 0.33
PIK3R1 P27986 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11254135 0.84 KIF11 (0.39) KIF11S1PR1S1PR3TRPV1GCGR
SCHEMBL28506866 0.83 KIF11 (0.38) KIF11S1PR1S1PR3GCGRNPC1
SCHEMBL7272903 0.79 PDE3B (0.44) GCGRMAPK14NPC1RAB9AHTT
SCHEMBL11231069 0.78 CYP2C19 (0.50) KIF11MAPK14LMNAHPGDTSHR
SCHEMBL11235418 0.76 RAB9A (0.43) TRPV1NPC1RAB9AMAPTLMNA
SCHEMBL11158174 0.76 CASP1 (0.51) MAPT
SCHEMBL7278230 0.75 PIK3R1 (0.36) GCGRMAPK14NPC1RAB9AHTT
SCHEMBL11173175 0.73 KIF11 (0.41) KIF11S1PR1S1PR3TRPV1GCGR
SCHEMBL11248447 0.72 SMN1; SMN2 (0.40) S1PR1GCGRMAPK14NPC1RAB9A
SCHEMBL21339368 0.71 PTGS2 (0.49) KIF11GCGRMAPK14NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4351941-A Pyridinyl-pyridines STERLING DRUG INC. (US) 1982-09-28 US disclosed
US-4331672-A 5-(Pyridinyl)pyridine-2-hydrazines, their preparation and their cardiotonic use STERLING DRUG INC. (US) 1982-05-25 US disclosed