SCHEMBL7278230

SCHEMBL7278230

CC(C)c1nc(Cl)c(Br)cc1-c1ccncc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3R1 P27986 1/20 0.36
PIK3CA P42336 1/20 0.36
GCGR P47871 4/20 0.35
MAPK14 Q16539 4/20 0.35
MAPK10 P53779 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.34
GSK3B P49841 2/20 0.34
HTT P42858 1/20 0.34
MAPK1 P28482 1/20 0.33
NPC1 O15118 3/20 0.32
RAB9A P51151 3/20 0.32
AKR1C3 P42330 1/20 0.32
AKR1C2 P52895 1/20 0.32
IMPDH2 P12268 1/20 0.32
AKT1 P31749 1/20 0.32
MAPT P10636 1/20 0.32
GFER P55789 1/20 0.32
ADORA2B P29275 2/20 0.31
NQO2 P16083 1/20 0.31
ADORA2A P29274 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11239183 0.84 GCGR (0.36) GCGRMAPK14MAPK10SMN1; SMN2GSK3B
SCHEMBL7272675 0.79 SQOR (0.40) PIK3R1PIK3CASMN1; SMN2NPC1RAB9A
SCHEMBL7272903 0.79 PDE3B (0.44) PIK3R1PIK3CAGCGRMAPK14SMN1; SMN2
SCHEMBL11232696 0.78 CYP2C19 (0.50) PIK3CAGSK3BHTT
SCHEMBL11155642 0.76 CASP1 (0.51) MAPTCCNCCDK8
SCHEMBL11233810 0.76 PDE7A (0.43) NPC1RAB9AMAPT
SCHEMBL11241215 0.75 KIF11 (0.37) PIK3R1PIK3CAGCGRMAPK14SMN1; SMN2
SCHEMBL11172843 0.73 RAB9A (0.37) GCGRMAPK14MAPK10SMN1; SMN2GSK3B
SCHEMBL11248447 0.72 SMN1; SMN2 (0.40) GCGRMAPK14SMN1; SMN2GSK3BHTT
SCHEMBL11389347 0.71 CASP1 (0.58) GCGRMAPK14GSK3BMAPK1IMPDH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4463008-A 2-Alkoxy-5-(pyridinyl)pyridines and cardiotonic use thereof STERLING DRUG INC. (US) 1984-07-31 US disclosed
EP-0109027-A1 Pyridine derivatives, process for their preparation and composition containing them STERLING DRUG INC. (US) 1984-05-23 EP disclosed
US-4351941-A Pyridinyl-pyridines STERLING DRUG INC. (US) 1982-09-28 US disclosed
US-4331672-A 5-(Pyridinyl)pyridine-2-hydrazines, their preparation and their cardiotonic use STERLING DRUG INC. (US) 1982-05-25 US disclosed