SCHEMBL11248404

SCHEMBL11248404

CN1CCC(C(=O)O)(c2ccccc2Sc2ccc(F)cc2)CC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.43
KDM4E B2RXH2 4/20 0.43
NPY1R P25929 1/20 0.43
NPY2R P49146 1/20 0.43
ALDH1A1 P00352 6/20 0.42
MAPT P10636 1/20 0.42
OPRM1 P35372 3/20 0.42
SLC6A9 P48067 2/20 0.41
L3MBTL1 Q9Y468 2/20 0.39
SLC22A1 O15245 1/20 0.39
SLC6A4 P31645 1/20 0.39
ADRA1A P35348 1/20 0.39
OPRD1 P41143 1/20 0.39
OPRK1 P41145 1/20 0.39
KCNH2 Q12809 1/20 0.39
GLA P06280 1/20 0.39
HTR1A P08908 1/20 0.39
HTR3A P46098 1/20 0.39
TDP1 Q9NUW8 1/20 0.38
CHRNA7 P36544 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11248843 0.88 ALDH1A1 (0.42) SMN1; SMN2ALDH1A1SLC6A9L3MBTL1GLA
SCHEMBL11258115 0.88 RHEB (0.44) SMN1; SMN2KDM4ENPY1RNPY2RALDH1A1
SCHEMBL11249097 0.82 HTR1A (0.46) SMN1; SMN2ALDH1A1OPRM1SLC6A9L3MBTL1
SCHEMBL11248413 0.82 SLC6A9 (0.43) SMN1; SMN2KDM4ENPY1RNPY2RALDH1A1
SCHEMBL11483187 0.82 SMN1; SMN2 (0.46) SMN1; SMN2KDM4ENPY1RNPY2RALDH1A1
Bromide SCHEMBL11427938 0.81 HTR1A (0.45) SMN1; SMN2ALDH1A1OPRM1SLC6A9L3MBTL1
Oxalic Acid SCHEMBL11487121 0.80 KDM4E (0.50) SMN1; SMN2KDM4ENPY1RNPY2RALDH1A1
SCHEMBL11477255 0.80 KDM4E (0.53) SMN1; SMN2KDM4EALDH1A1MAPTOPRM1
SCHEMBL11482078 0.80 SMN1; SMN2 (0.44) SMN1; SMN2KDM4ENPY1RNPY2RALDH1A1
SCHEMBL11477977 0.79 SMN1; SMN2 (0.46) SMN1; SMN2KDM4ENPY1RNPY2RALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4198419-A Phenylthiophenylpiperidines AMERICAN HOECHST CORPORATION (US) 1980-04-15 US claimed
EP-0013424-B1 SPIRO(DIBENZO(B,F)THIEPINE-PIPERIDINES), INTERMEDIATE PRODUCTS FOR THEIR PREPARATION AND MEDICAMENTS CONTAINING THEM HOECHST AKTIENGESELLSCHAFT (DE) 1982-11-17 EP disclosed
EP-0013424-A1 Spiro(dibenzo(b,f)thiepine-piperidines), intermediate products for their preparation and medicaments containing them HOECHST AKTIENGESELLSCHAFT (DE) 1980-07-23 EP disclosed
US-4198420-A Spiro[dibenz(b,f)thiepin-piperidine]s AMERICAN HOECHST CORPORATION (US) 1980-04-15 US disclosed
US-4198419-A Phenylthiophenylpiperidines AMERICAN HOECHST CORPORATION (US) 1980-04-15 US disclosed